SCHEMBL9213545

SCHEMBL9213545

Cc1ccc(S(=O)(=O)N2CCC[C@@]2(O)C(=O)O)cc1

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CYP2C19 P33261 1/20 0.53
ALDH1A1 P00352 4/20 0.46
PKM P14618 3/20 0.46
POLB P06746 1/20 0.46
HTT P42858 1/20 0.46
HPGD P15428 1/20 0.44
NPSR1 Q6W5P4 1/20 0.44
KMT2A Q03164 6/20 0.43
GAA P10253 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
MEN1 O00255 4/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
USP2 O75604 1/20 0.42
LMNA P02545 1/20 0.42
NPC1 O15118 1/20 0.42
RAB9A P51151 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8206367 0.85 HSD11B1 (0.57) ALDH1A1PKMPOLBHTTKMT2A
SCHEMBL9208624 0.85 PKM (0.46) CYP2C19ALDH1A1PKMPOLBHTT
SCHEMBL7407681 0.83 CYP2C19 (0.56) CYP2C19ALDH1A1PKMPOLBHTT
SCHEMBL10905546 0.83 ALDH1A1 (0.41) CYP2C19ALDH1A1PKMPOLBHTT
SCHEMBL18221902 0.77 CYP2C19 (0.53) CYP2C19ALDH1A1PKMPOLBHTT
SCHEMBL9217072 0.77 KMT2A (0.47) CYP2C19ALDH1A1PKMPOLBHTT
SCHEMBL7250447 0.77 CYP2C19 (0.59) CYP2C19ALDH1A1PKMPOLBHTT
SCHEMBL18221869 0.76 CYP2C19 (0.52) CYP2C19ALDH1A1PKMPOLBHTT
SCHEMBL11888884 0.74 CYP2C19 (0.67) CYP2C19ALDH1A1PKMPOLBHTT
SCHEMBL8199043 0.73 MMP1 (0.52) ALDH1A1PKMPOLBHTTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0345808-B1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines BRISTOL MYERS SQUIBB CO (US) 1995-01-11 EP disclosed
EP-0400661-A1 Agents for treatment of brain ischemia Bristol-Myers Squibb Company (US) 1990-12-05 EP disclosed
US-4954502-A Antidepressants BRISTOL-MYERS SQUIBB COMPANY (US) 1990-09-04 US disclosed
EP-0345808-A1 1-Indolylalkyl-4-(substituted-pyridinyl)piperazines Bristol-Myers Squibb Company (US) 1989-12-13 EP disclosed
US-3951980-A 3-Substituted-8-methyl-3,8-diazabicyclo[3.2.1]octanes STANFORD RESEARCH INSTITUTE (US) 1976-04-20 US disclosed
US-3947445-A Diazabicyclooctanes and diazabicycloheptanes STANFORD RESEARCH INSTITUTE (US) 1976-03-30 US disclosed