SCHEMBL9214121

SCHEMBL9214121

Cc1cc2c(cc1C)CN(CC1CCN(Cc3cccnc3)C1)C2

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CHRNB2 P17787 1/20 0.46
CHRNA4 P43681 1/20 0.46
CACNA1I Q9P0X4 1/20 0.44
KDM4E B2RXH2 2/20 0.43
PDE2A O00408 1/20 0.43
TRPV6 Q9H1D0 2/20 0.43
CHRM2 P08172 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42
ALDH1A1 P00352 1/20 0.42
MAPT P10636 1/20 0.42
HTT P42858 1/20 0.42
MAPK1 P28482 1/20 0.41
KMT2A Q03164 2/20 0.41
GFER P55789 1/20 0.40
PTGER2 P43116 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9214611 0.88 PTGER2 (0.48) KDM4ECHRM2CHRM1CHRM3GFER
SCHEMBL9217159 0.81 ACHE (0.44) CHRNB2CHRNA4CACNA1IKDM4EPDE2A
Hydrochloric Acid SCHEMBL9206800 0.79 DRD2 (0.41) CHRNB2CHRNA4CACNA1IKDM4EALDH1A1
SCHEMBL9206955 0.77 DRD2 (0.44) CHRNB2CHRNA4CACNA1IKDM4EPDE2A
SCHEMBL803678 0.77 CHRNB2 (0.54) CHRNB2CHRNA4CACNA1IKDM4ETRPV6
SCHEMBL23291216 0.76 CHRNB2 (0.56) CHRNB2CHRNA4CACNA1IKDM4ETRPV6
SCHEMBL9211536 0.76 CHRNB2 (0.56) CHRNB2CHRNA4CACNA1IKDM4ETRPV6
SCHEMBL23291215 0.76 CHRNB2 (0.56) CHRNB2CHRNA4CACNA1IKDM4ETRPV6
SCHEMBL9216662 0.75 HRH3 (0.43)
Hydrochloric Acid SCHEMBL9216765 0.75 HRH3 (0.41) CHRM2CHRM1CHRM3KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed