SCHEMBL9217159

SCHEMBL9217159

Cc1cc2c(cc1C)C(=O)N(CC1CCN(Cc3cccnc3)C1)CC2

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.44
CACNA1I Q9P0X4 1/20 0.40
KDM4E B2RXH2 2/20 0.40
DHPS P49366 1/20 0.40
TRPV6 Q9H1D0 1/20 0.39
ALDH1A1 P00352 2/20 0.39
CHRNB2 P17787 1/20 0.39
CHRNA4 P43681 1/20 0.39
MAPT P10636 1/20 0.39
HTT P42858 1/20 0.39
PARP1 P09874 2/20 0.38
PARP2 Q9UGN5 2/20 0.38
GRM5 P41594 1/20 0.38
PDE2A O00408 1/20 0.38
MAPK1 P28482 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
TDP1 Q9NUW8 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9213558 0.86 ACHE (0.42) ACHECACNA1IALDH1A1MAPTKMT2A
Hydrochloric Acid SCHEMBL9213433 0.85 ACHE (0.41) ACHECACNA1IALDH1A1MAPTKMT2A
SCHEMBL9214452 0.84 GRM5 (0.40) CHRNB2CHRNA4GRM5
SCHEMBL9215804 0.83 GRM5 (0.39) KDM4ECHRNB2CHRNA4GRM5KMT2A
Hydrochloric Acid SCHEMBL9214335 0.83 GRM5 (0.39) CHRNB2CHRNA4GRM5
SCHEMBL9214121 0.81 CHRNB2 (0.46) CACNA1IKDM4ETRPV6ALDH1A1CHRNB2
SCHEMBL9215061 0.80 ACHE (0.46) ACHEKDM4E
SCHEMBL9213007 0.79 GRM5 (0.38) ACHEGRM5
Hydrochloric Acid SCHEMBL9216230 0.78 GRM5 (0.37) ACHEGRM5
SCHEMBL9215461 0.76 BCHE (0.56) ACHEKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed
EP-0292840-A2 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation Dr. Karl Thomae GmbH (DE) 1988-11-30 EP disclosed