SCHEMBL9206955

SCHEMBL9206955

c1cncc(CN2CCC(CN3CCc4cc5c(cc4CC3)OCO5)C2)c1

nearest known ligand 0.44

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.44
KCNH2 Q12809 1/20 0.44
KDM4E B2RXH2 4/20 0.43
ALDH1A1 P00352 2/20 0.43
MAPT P10636 2/20 0.43
CHRNB2 P17787 1/20 0.43
CHRNA4 P43681 1/20 0.43
GAA P10253 1/20 0.43
MCHR1 Q99705 1/20 0.43
CACNA1I Q9P0X4 1/20 0.42
TDP1 Q9NUW8 1/20 0.41
UBE2M P61081 1/20 0.41
DCUN1D1 Q96GG9 1/20 0.41
POLB P06746 1/20 0.40
HTT P42858 1/20 0.40
MEN1 O00255 1/20 0.40
LMNA P02545 1/20 0.40
KMT2A Q03164 1/20 0.40
PDE2A O00408 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9206800 0.95 DRD2 (0.41) DRD2KCNH2KDM4EALDH1A1MAPT
SCHEMBL9213558 0.86 ACHE (0.42) ALDH1A1MAPTMCHR1CACNA1ITDP1
Hydrochloric Acid SCHEMBL9213433 0.84 ACHE (0.41) ALDH1A1MAPTMCHR1CACNA1ITDP1
Hydrochloric Acid SCHEMBL9204880 0.78 CCR2 (0.38) KCNH2KDM4ECHRNB2CHRNA4MEN1
SCHEMBL9215978 0.77 PDE5A (0.39)
SCHEMBL9214121 0.77 CHRNB2 (0.46) KDM4EALDH1A1MAPTCHRNB2CHRNA4
SCHEMBL9739331 0.76 MEN1 (0.47) KCNH2KDM4EALDH1A1MEN1LMNA
Hydrochloric Acid SCHEMBL9213791 0.75 ACHE (0.37)
SCHEMBL9214611 0.74 PTGER2 (0.48) KDM4E
SCHEMBL23291215 0.74 CHRNB2 (0.56) KDM4EALDH1A1MAPTCHRNB2CHRNA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0292840-B1 Cyclic amine derivatives, medicaments containing these compounds and procedure for their preparation THOMAE GMBH DR K (DE) 1995-08-09 EP disclosed
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed