SCHEMBL9740563

SCHEMBL9740563

O=C1Cc2cc3c(cc2CCN1CC1CCCNC1)OOC3

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 1/20 0.39
PARP1 P09874 1/20 0.36
NAAA Q02083 1/20 0.34
CDK9 P50750 2/20 0.33
GRM5 P41594 1/20 0.31
KHK P50053 1/20 0.31
CCR2 P41597 1/20 0.31
KCNH2 Q12809 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9740567 0.85 DRD2 (0.41) DRD2PARP1NAAACDK9GRM5
SCHEMBL9207567 0.82 DRD2 (0.39) DRD2PARP1NAAACDK9GRM5
SCHEMBL9740217 0.81 ITGB3 (0.39) DRD2PARP1CDK9GRM5KHK
SCHEMBL9212186 0.79 SMN1; SMN2 (0.48) DRD2PARP1KCNH2
SCHEMBL9215737 0.78 DRD2 (0.40) DRD2PARP1NAAACDK9GRM5
SCHEMBL9204902 0.76 SMN1; SMN2 (0.47) DRD2KCNH2
SCHEMBL9739351 0.74 ITGB3 (0.36) DRD2PARP1CDK9GRM5KHK
SCHEMBL9740805 0.74 PARP1 (0.45) DRD2PARP1GRM5KHK
SCHEMBL9205660 0.72 GRM5 (0.42) DRD2PARP1CDK9GRM5
SCHEMBL9213734 0.69 GRM5 (0.41) DRD2PARP1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5175157-A Cardiovascular disorders BOEHRINGER INGELHEIM GMBH (DE) 1992-12-29 US disclosed