Iodide

Iodide

SCHEMBL9218396

CC(C)(C)OC(=O)C[C@H](NC(=O)CC(=O)NCCc1ccc(C(=N)N)cc1)C(=O)N[C@@H](Cc1ccccc1)C(=O)OC(C)(C)C.I

nearest known ligand 0.47

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHECHRM1CHRM3CHRNA1CHRNB1CHRNDCHRNECHRNG

The experimentally established mechanism targets of Iodide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ST14 Q9Y5Y6 2/20 0.47
F10 P00742 1/20 0.44
MMP1 P03956 2/20 0.44
MMP3 P08254 2/20 0.44
MMP9 P14780 1/20 0.44
CA2 P00918 1/20 0.43
ITGB3 P05106 2/20 0.43
ITGA2B P08514 2/20 0.43
REN P00797 2/20 0.42
PRSS1 P07477 1/20 0.42
TMPRSS15 P98073 1/20 0.42
MAPT P10636 2/20 0.41
TDP1 Q9NUW8 2/20 0.41
TMPRSS11D O60235 1/20 0.41
KLK5 Q9Y337 1/20 0.40
MMP8 P22894 1/20 0.40
F7 P08709 2/20 0.39
ADRA1B P35368 1/20 0.39
CTSL P07711 1/20 0.39
POLB P06746 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9218412 0.99 ST14 (0.47) ST14F10MMP1MMP3MMP9
Iodide SCHEMBL9217545 0.88 CCKBR (0.42) F10MMP1MMP3MMP9ITGB3
Iodide SCHEMBL9221941 0.86 CCKBR (0.43) F10MMP1MMP3MMP9ITGB3
SCHEMBL7338218 0.85 CTSS (0.45) MMP1MMP3MMP9CA2MAPT
SCHEMBL7296817 0.85 MAPT (0.44) F10MMP1MMP3MMP9ITGB3
SCHEMBL9217556 0.83 REN (0.49) RENTMPRSS11DKLK5
Iodide SCHEMBL9215204 0.82 ITGB3 (0.51) MMP1MMP3MMP9ITGB3ITGA2B
SCHEMBL9215140 0.81 REN (0.47) F10MMP1MMP3MMP9REN
SCHEMBL9215215 0.81 ITGB3 (0.52) MMP1MMP3MMP9ITGB3ITGA2B
Iodide SCHEMBL9866079 0.80 MAPT (0.43) F10ITGB3ITGA2BPRSS1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5430024-A Peptides bearing N-terminal amidino moieties and their use as inhibitors of platelet aggregation HOFFMANN-LA ROCHE INC. (US) 1995-07-04 US disclosed
US-5273982-A An amidinoaryleneamidoalkylpiperazinyleneacetic acid HOFFMANN-LA ROCHE INC. (US) 1993-12-28 US disclosed