SCHEMBL9218534

SCHEMBL9218534

Oc1cccc(-c2cnn3c(O)ncnc23)c1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRC P12931 7/20 0.47
KDR P35968 5/20 0.47
LCK P06239 4/20 0.47
HCK P08631 3/20 0.47
PIK3CG P48736 3/20 0.44
PIK3CD O00329 2/20 0.44
PIK3CA P42336 2/20 0.44
PIK3CB P42338 2/20 0.44
PRKDC P78527 2/20 0.44
HSD17B1 P14061 2/20 0.44
HSD17B2 P37059 2/20 0.44
ABL1 P00519 4/20 0.42
EGFR P00533 3/20 0.42
ABL2 P42684 2/20 0.42
JAK2 O60674 2/20 0.42
NTRK1 P04629 2/20 0.42
INSR P06213 2/20 0.42
NPM1 P06748 2/20 0.42
CSF1R P07333 2/20 0.42
LYN P07948 2/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9219234 0.86 NPC1 (0.57) SRCKDRABL1EGFRABL2
SCHEMBL9212913 0.86 EGLN2 (0.43) SRCKDRLCKHCKMEN1
SCHEMBL9221803 0.86 ALDH1A1 (0.44) SRCKDRLCKHCKMEN1
SCHEMBL9172768 0.84 RAB9A (0.55) KDRMEN1NPC1RAB9AKMT2A
SCHEMBL9214289 0.82 KDR (0.50) SRCKDRABL1EGFRABL2
SCHEMBL9216208 0.82 SMN1; SMN2 (0.40) SRCKDRLCKHCKNTRK1
SCHEMBL9215756 0.81 SRC (0.45) SRCKDRLCKHCKABL1
SCHEMBL9212121 0.81 KDR (0.44) SRCKDRLCKPIK3CGPIK3CD
SCHEMBL9221859 0.81 CYP17A1 (0.45) SRCKDRHCKPIK3CGPIK3CD
SCHEMBL9221094 0.80 MAPT (0.43) PIK3CGPIK3CDPIK3CAPIK3CBPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0269859-B2 Pyrazolotriazine compounds OTSUKA PHARMA CO LTD (JP) 1995-10-18 EP disclosed
US-4824834-A TREATING GOUT OTSUKA PHARMACEUTICAL COMPANY, LIMITED (JP) 1989-04-25 US disclosed
EP-0269859-A2 Pyrazolotriazine compounds OTSUKA PHARMACEUTICAL CO., LTD. (JP) 1988-06-08 EP disclosed