SCHEMBL9219903

SCHEMBL9219903

COC(=O)C(Cl)C(=O)c1ccc(F)c(F)c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRNA1 P02708 1/20 0.55
CHRNG P07510 1/20 0.55
CHRNB1 P11230 1/20 0.55
CHRNB2 P17787 1/20 0.55
SLC6A2 P23975 1/20 0.55
CHRNB4 P30926 1/20 0.55
CHRNA3 P32297 1/20 0.55
CHRNA4 P43681 1/20 0.55
SLC6A3 Q01959 1/20 0.55
CHRND Q07001 1/20 0.55
CES2 O00748 2/20 0.49
CES1 P23141 2/20 0.49
SMN1; SMN2 Q16637 2/20 0.44
GAA P10253 1/20 0.44
MEN1 O00255 5/20 0.40
KMT2A Q03164 5/20 0.40
POLB P06746 1/20 0.40
KCNQ3 O43525 3/20 0.39
KCNQ2 O43526 3/20 0.39
RAB9A P51151 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8875867 0.88 KCNQ3 (0.43) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL29037468 0.86 KCNQ3 (0.42) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL9221209 0.84 CES2 (0.46) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL9219929 0.82 CES2 (0.44) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL1533349 0.81 RAB9A (0.44) CES2CES1SMN1; SMN2GAAMEN1
SCHEMBL9227046 0.81 CHRNA1 (0.58) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL7500254 0.81 CHRNA1 (0.55) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL9745320 0.80 ESR1 (0.42) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL9226597 0.80 CES2 (0.54) CHRNA1CHRNGCHRNB1CHRNB2SLC6A2
SCHEMBL9431238 0.80 MEN1 (0.49) CES2CES1SMN1; SMN2GAAMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0303291-B1 Fluorinated benzoyl compounds ASAHI GLASS CO LTD (JP) 1995-04-26 EP disclosed
US-5093515-A Intermediate for quinolone carboxylic acid bactericide ASAHI GLASS COMPANY LTD. (JP) 1992-03-03 US disclosed
US-5068449-A FLUORINATED BENZOYL COMPOUNDS ASAHI GLASS COMPANY, LTD. (JP) 1991-11-26 US disclosed
EP-0303291-A2 Fluorinated benzoyl compounds ASAHI GLASS COMPANY LTD. (JP) 1989-02-15 EP disclosed