SCHEMBL9220779

SCHEMBL9220779

COCCOC(=O)OC1=C(C)N(C)C(C)=C(OC(=O)OC(C)C)C1c1ccc(C#N)cc1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA2A P08913 1/20 0.35
ADRA2B P18089 1/20 0.35
ADRA2C P18825 1/20 0.35
ADRA1D P25100 1/20 0.35
ADRA1A P35348 1/20 0.35
ADRA1B P35368 1/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
CYP1A2 P05177 2/20 0.35
CYP3A4 P08684 2/20 0.35
CYP2C9 P11712 2/20 0.35
CYP2C19 P33261 2/20 0.35
LMNA P02545 2/20 0.35
TSHR P16473 2/20 0.35
CYP2D6 P10635 1/20 0.35
NFKB1 P19838 1/20 0.35
THPO P40225 1/20 0.35
MAPT P10636 1/20 0.35
HTT P42858 3/20 0.34
CACNA1F O60840 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9222084 0.87 CACNA1F (0.41) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9214880 0.87 HPGD (0.46) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9364254 0.84 HSP90AA1 (0.40) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9364303 0.83 HPGD (0.40) CYP3A4CYP2C9TSHRHTTHPGD
SCHEMBL9215408 0.83 KDM4E (0.37) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9220053 0.82 HTT (0.48) ADRA2AADRA2BADRA2CADRA1DADRA1A
SCHEMBL10913259 0.77 CACNA1C (0.55) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9220730 0.77 APOBEC3A (0.36) MEN1KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL9364248 0.76 HSP90AA1 (0.44) KMT2ALMNATSHRMAPTHTT
SCHEMBL9222124 0.76 PYGM (0.37) MEN1KMT2ACYP1A2CYP3A4CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525568-B1 N-Alkylated 1,4-dihydropyridine carboxylicacid ester derivatives BAYER AG (DE) 1995-05-10 EP claimed
EP-0525568-A1 N-Alkylated 1,4-dihydropyridine carboxylicacid ester derivatives BAYER AG (DE) 1993-02-03 EP claimed
EP-0525568-B1 N-Alkylated 1,4-dihydropyridine carboxylicacid ester derivatives BAYER AG (DE) 1995-05-10 EP disclosed
EP-0525568-A1 N-Alkylated 1,4-dihydropyridine carboxylicacid ester derivatives BAYER AG (DE) 1993-02-03 EP disclosed