SCHEMBL9230253

SCHEMBL9230253

CN1CCN(c2cccc3c(=O)n(-c4ccc(Cl)cc4)cnc23)CC1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 1/20 0.51
WEE1 P30291 4/20 0.43
MCHR1 Q99705 1/20 0.42
TRPV4 Q9HBA0 2/20 0.41
ABCB1 P08183 1/20 0.41
DRD2 P14416 2/20 0.41
DRD3 P35462 2/20 0.41
ALDH1A1 P00352 2/20 0.41
GRM1 Q13255 2/20 0.41
MAPT P10636 1/20 0.41
ALOX12 P18054 1/20 0.41
HTR1A P08908 1/20 0.40
DRD4 P21917 1/20 0.40
HTR2A P28223 1/20 0.40
HTR2C P28335 1/20 0.40
USP2 O75604 1/20 0.40
CYP1A2 P05177 1/20 0.40
GLA P06280 1/20 0.40
CYP3A4 P08684 1/20 0.40
CASP1 P29466 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1040982 0.78 TRPV4 (0.50) TRPV4ALDH1A1GRM1CYP1A2CYP3A4
SCHEMBL4827730 0.76 MAPK14 (0.45) USP2CASP1CASP7
SCHEMBL20886963 0.69 RAB9A (1.00) RAB9ADRD2DRD3MAPTHTR1A
SCHEMBL5256633 0.68 MCHR1 (0.73) MCHR1DRD3HTR2CCYP3A4
SCHEMBL5429660 0.66 GRM1 (0.52) RAB9AGRM1GRM5
SCHEMBL8245138 0.66 GRM1 (0.60) RAB9AALDH1A1GRM1GRM5
SCHEMBL23131531 0.66 DRD2 (0.46) DRD2DRD3ALDH1A1MAPTHTR1A
SCHEMBL28311804 0.65 ADRA2C (0.53) DRD2DRD3MAPT
SCHEMBL8247056 0.65 GRM1 (0.78) ALDH1A1GRM1GRM5
SCHEMBL8245805 0.65 GRM1 (0.74) ALDH1A1GRM1GRM5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-7258224-A None JP disclosed
JP-H07258224-A BICYCLIC COMPOUND DAI ICHI SEIYAKU CO LTD 1995-10-09 JP disclosed