SCHEMBL9230332

SCHEMBL9230332

CCOC(=O)CN1C(=O)C(NC(=O)[C@H](Cc2ccccc2)SC(C)=O)C=Cc2ccccc21

nearest known ligand 0.43

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCKBR P32239 3/20 0.38
CCKAR P32238 1/20 0.38
HRH4 Q9H3N8 1/20 0.38
ACE P12821 4/20 0.37
MME P08473 3/20 0.37
LMNA P02545 2/20 0.36
ALDH1A1 P00352 1/20 0.36
PPARG P37231 1/20 0.36
PPARA Q07869 1/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
NPSR1 Q6W5P4 1/20 0.35
ABCB11 O95342 1/20 0.35
AGTR2 P50052 1/20 0.35
PDE3A Q14432 1/20 0.35
TDP1 Q9NUW8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9228780 0.90 CCKBR (0.39) CCKBRCCKARHRH4ACESMN1; SMN2
SCHEMBL9226683 0.84 LMNA (0.36) CCKBRCCKARLMNAALDH1A1SMN1; SMN2
SCHEMBL7439940 0.79 ACE (0.59) ACEMMEABCB11AGTR2PDE3A
SCHEMBL7439947 0.79 ACE (0.59) ACEMMEABCB11AGTR2PDE3A
SCHEMBL9230696 0.78 CCKBR (0.39) CCKBRCCKARLMNAALDH1A1SMN1; SMN2
SCHEMBL11118972 0.76 NFKB1 (0.46) CCKBRCCKARLMNAALDH1A1SMN1; SMN2
SCHEMBL9227099 0.74 ACE (0.59) ACEMME
SCHEMBL8881603 0.73 LMNA (0.49) CCKBRCCKARLMNAALDH1A1SMN1; SMN2
SCHEMBL10498972 0.73 LMNA (0.49) CCKBRCCKARLMNAALDH1A1SMN1; SMN2
SCHEMBL9228102 0.71 P2RX4 (0.40) LMNAALDH1A1SMN1; SMN2NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0671172-A1 AMINO ACID DERIVATIVE Eisai Co., Ltd. (JP) 1995-09-13 EP disclosed