SCHEMBL9230358

SCHEMBL9230358

CCCNc1cc2cccc(N3CCNCC3)c2oc1=O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BACE1 P56817 4/20 0.44
HTR1A P08908 2/20 0.41
HTR2A P28223 2/20 0.41
DRD2 P14416 1/20 0.41
DRD4 P21917 1/20 0.41
HTR2C P28335 1/20 0.41
DRD3 P35462 1/20 0.41
HTR6 P50406 2/20 0.40
HTR5A P47898 2/20 0.40
HTR3E A5X5Y0 1/20 0.40
HTR3B O95264 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
NCF1 P14598 1/20 0.40
TSHR P16473 1/20 0.40
NFKB1 P19838 1/20 0.40
HTR1D P28221 1/20 0.40
HTR1B P28222 1/20 0.40
HTR7 P34969 1/20 0.40
MTOR P42345 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9230841 0.84 BACE1 (0.48) BACE1HTR1AHTR2AHTR2CHTR6
Hydrochloric Acid SCHEMBL9230054 0.83 BACE1 (0.47) BACE1HTR1AHTR2AHTR2CHTR6
SCHEMBL9227350 0.82 DRD2 (0.50) BACE1HTR1ADRD2DRD4DRD3
SCHEMBL929137 0.81 KDM4E (0.54) BACE1HTR6HTR5ACYP1A2HSD17B10
SCHEMBL9274710 0.80 HTR1A (0.47) BACE1HTR1AHTR2ADRD2DRD4
SCHEMBL9229904 0.78 ADRB1 (0.51) BACE1HTR1AHTR2AHTR6HTR5A
Hydrochloric Acid SCHEMBL9229290 0.77 ADRB1 (0.50) BACE1HTR1AHTR2AHTR6HTR5A
SCHEMBL9228925 0.76 HTR5A (0.52) BACE1HTR1AHTR2AHTR2CHTR6
Hydrochloric Acid SCHEMBL9225164 0.75 HTR5A (0.51) BACE1HTR1AHTR2AHTR2CHTR6
SCHEMBL9229724 0.75 HTR6 (0.48) BACE1HTR1AHTR2ADRD2HTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-1105360-A 1-[2H-1-benzopyran-2-one-8yl]-piperazin derivative DUPHAR INT RES (NL) 1995-07-19 CN disclosed
EP-0650964-A1 1 2H-1-benzopyran-2-one-8-yl -piperazine derivatives DUPHAR INTERNATIONAL RESEARCH B.V (NL) 1995-05-03 EP disclosed