SCHEMBL9230707

SCHEMBL9230707

O=C1Nc2cccnc2C2(c3cccc(Cl)c3)OCCN12

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 1/20 0.38
HTR1A P08908 1/20 0.37
HTR2A P28223 1/20 0.37
HTR7 P34969 1/20 0.37
HTR6 P50406 1/20 0.37
GHSR Q92847 1/20 0.35
PGR P06401 4/20 0.35
BRD4 O60885 1/20 0.34
OPRL1 P41146 1/20 0.34
MEN1 O00255 1/20 0.33
CYP1A2 P05177 1/20 0.33
MAPT P10636 1/20 0.33
HPGD P15428 1/20 0.33
CYP2C19 P33261 1/20 0.33
KMT2A Q03164 1/20 0.33
TRPA1 O75762 2/20 0.33
PKLR P30613 1/20 0.33
CHRNA1 P02708 2/20 0.33
CHRNG P07510 2/20 0.33
CHRNB1 P11230 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9231150 0.88 OPRL1 (0.35) OPRL1MEN1CYP1A2MAPTCYP2C19
SCHEMBL9230320 0.86 OPRL1 (0.38) BRD4OPRL1CYP1A2OTUD7B
SCHEMBL9225503 0.83 AKR1C3 (0.47) AKR1C3HTR1AHTR2AHTR7HTR6
SCHEMBL9043134 0.78 MAPT (0.36) HTR1AHTR2AHTR7HTR6GHSR
SCHEMBL9231680 0.76 CCR1 (0.33) OPRL1CYP1A2MAPTCYP2C19OTUD7B
SCHEMBL9231434 0.76 L3MBTL1 (0.34) PKLROTUD7B
SCHEMBL11869473 0.74 AKR1C3 (0.51) AKR1C3HTR1AHTR2AHTR7HTR6
SCHEMBL9232012 0.74 AKR1C3 (0.56) AKR1C3HTR1AHTR2AHTR7HTR6
SCHEMBL9231114 0.72 AKR1C3 (0.42) AKR1C3HTR1AHTR2AHTR7HTR6
SCHEMBL9230546 0.72 LMNA (0.43) AKR1C3BRD4OPRL1MEN1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0640087-A1 USE OF TRICYCLIC PYRIMIDINE DERIVATIVES AS ANTI-VIRAL MEDICAMENTS Roche Diagnostics GmbH (DE) 1995-03-01 EP disclosed
WO-1993023405-A1 USE OF TRICYCLIC PYRIMIDINE DERIVATIVES AS ANTI-VIRAL MEDICAMENTS BOEHRINGER MANNHEIM GMBH (DE) 1993-11-25 WO disclosed