SCHEMBL9230726

SCHEMBL9230726

CN(C)CCOc1ccc(-c2nn(CCN(C)C)c3ncccc23)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 1/20 0.42
CHRNB2 P17787 1/20 0.42
CHRNA4 P43681 1/20 0.42
PTPN1 P18031 1/20 0.41
TNK2 Q07912 1/20 0.41
LTA4H P09960 2/20 0.41
TNKS O95271 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
CYP2C19 P33261 1/20 0.40
LSS P48449 1/20 0.40
ADORA3 P0DMS8 1/20 0.40
ADORA2A P29274 1/20 0.40
ADORA2B P29275 1/20 0.40
ADORA1 P30542 1/20 0.40
ACHE P22303 1/20 0.40
PAX8 Q06710 1/20 0.39
KAT2B Q92831 1/20 0.39
KDM4E B2RXH2 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9234490 0.90 GSK3B (0.50) GSK3BPTPN1CYP1A2CYP2D6CYP2C9
SCHEMBL9876938 0.87 LSS (0.45) GSK3BPTPN1CYP1A2CYP2D6CYP2C9
Maleic Acid SCHEMBL9237612 0.84 LSS (0.40) GSK3BTNK2LSSACHEKDM4E
Fumaric Acid SCHEMBL9237617 0.84 LSS (0.40) GSK3BTNK2LSSACHEKDM4E
SCHEMBL9876891 0.83 LSS (0.44) GSK3BLTA4HLSSACHEKDM4E
SCHEMBL9876682 0.82 GSK3B (0.43) GSK3BPTPN1CYP2D6CYP2C9LSS
SCHEMBL9876736 0.82 GAA (0.49) KDM4EESR1
SCHEMBL9876810 0.82 TNK2 (0.46) CHRNB2CHRNA4PTPN1TNK2LTA4H
SCHEMBL9224007 0.81 LSS (0.44) GSK3BPTPN1CYP1A2CYP2D6CYP2C9
SCHEMBL9876863 0.81 ACHE (0.41) TNKSCYP1A2CYP2D6CYP2C9CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0641564-A1 OPTICALLY ACTIVE CONDENSED PYRAZOLE COMPOUND FOR USE IN TREATING THROMBOCYTOPENIA AND ERYTHROPENIA YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1995-03-08 EP disclosed
US-5006520-A Antibiotics, antitumor agents, treatment of blood disorders YOSHITOMI PHARMACEUTICAL INDUSTRIES, LTD. (JP) 1991-04-09 US disclosed
EP-0338087-A1 FUSED PYRAZOLE COMPOUNDS, PROCESS FOR THEIR PREPARATION, AND THEIR MEDICINAL USE Yoshitomi Pharmaceutical Industries, Ltd. (JP) 1989-10-25 EP disclosed