SCHEMBL9250026

SCHEMBL9250026

CS(=O)(=O)c1cc(C=O)cc(O)c1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
XDH P47989 1/20 0.44
KDM4E B2RXH2 1/20 0.41
PTGS2 P35354 1/20 0.41
RAB9A P51151 1/20 0.41
ALDH1A1 P00352 2/20 0.38
AOX1 Q06278 1/20 0.38
FNTA P49354 1/20 0.37
FNTB P49356 1/20 0.37
TRIM24 O15164 1/20 0.34
HPGD P15428 1/20 0.34
ALDH5A1 P51649 1/20 0.34
ABAT P80404 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
TRIM33 Q9UPN9 1/20 0.34
ESR1 P03372 1/20 0.34
ESR2 Q92731 1/20 0.34
EGFR P00533 1/20 0.33
GABBR2 O75899 1/20 0.33
GABBR1 Q9UBS5 1/20 0.33
WDR5 P61964 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15783652 0.82 XDH (0.46) XDHKDM4EPTGS2RAB9AALDH1A1
SCHEMBL8996225 0.79 ALDH1A1 (0.49) KDM4EPTGS2ALDH1A1AOX1TRIM24
SCHEMBL24038842 0.77 PTGS2 (0.55) XDHKDM4EPTGS2RAB9AALDH1A1
SCHEMBL30456577 0.77 PTGS2 (0.55) XDHKDM4EPTGS2RAB9AALDH1A1
SCHEMBL27935044 0.76 XDH (0.59) XDHKDM4EPTGS2RAB9AALDH1A1
SCHEMBL132439 0.76 XDH (0.59) XDHKDM4EPTGS2RAB9AALDH1A1
Water SCHEMBL36578 0.74 XDH (0.57) XDHKDM4EPTGS2RAB9AALDH1A1
SCHEMBL31122716 0.74 XDH (0.57) XDHKDM4EPTGS2RAB9AALDH1A1
SCHEMBL16309120 0.74 SELL (0.54) KDM4EALDH1A1TDP1ESR1ESR2
SCHEMBL9248011 0.72 CA1 (0.50) ALDH1A1HPGDWDR5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 46 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9622988-B2 Small molecule xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2017-04-18 US disclosed
US-9622988-B2 Small molecule xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2017-04-18 US disclosed
US-9610257-B2 Small molecule xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2017-04-04 US disclosed
US-9610257-B2 Small molecule xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2017-04-04 US disclosed
US-9585848-B2 Small molecule xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2017-03-07 US disclosed
US-9585848-B2 Small molecule xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2017-03-07 US disclosed
US-9585847-B2 Small molecule xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2017-03-07 US disclosed
US-9585847-B2 Small molecule xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2017-03-07 US disclosed
US-9580379-B2 Xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2017-02-28 US disclosed
US-9580379-B2 Xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2017-02-28 US disclosed
US-8883858-B1 Small molecule xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2014-11-11 US disclosed
US-8883857-B2 Small molecule xanthine oxidase inhibitors and methods of use BAYLOR COLLEGE OF MEDICINE (US) 2014-11-11 US disclosed
US-20140329909-A1 SMALL MOLECULE XANTHINE OXIDASE INHIBITORS AND METHODS OF USE BAYLOR COLLEGE OF MEDICINE 2014-11-06 US disclosed
US-20140329909-A1 SMALL MOLECULE XANTHINE OXIDASE INHIBITORS AND METHODS OF USE BAYLOR COLLEGE OF MEDICINE 2014-11-06 US disclosed
US-20140163045-A1 Small Molecule Xanthine Oxidase Inhibitors and Methods of Use BAYLOR COLLEGE OF MEDICINE (US) 2014-06-12 US disclosed
US-20140163045-A1 Small Molecule Xanthine Oxidase Inhibitors and Methods of Use BAYLOR COLLEGE OF MEDICINE (US) 2014-06-12 US disclosed
US-5446194-A Pharmacologically active catechol derivatives ORION-YHTYMA OY (FI) 1995-08-29 US disclosed
US-5283352-A Transferase inhibitor ORION-YHTYMA OY (FI) 1994-02-01 US disclosed
US-5112861-A Inhibitors of catechol-methyl-transferase enzyme, levodopa ORION-YHTYMA OY (FI) 1992-05-12 US disclosed
US-4963590-A ENZYME INHIBITOR FOR TREATING PARKINSON'S DISEASE ALONG WITH DOPA;POTENTIATION ORION-YHTYMA OY (FI) 1990-10-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140329909-A1 SMALL MOLECULE XANTHINE OXIDASE INHIBITORS AND METHODS OF USE XDH, PNPO, AOX1 XDH 1/4885KDM4E 3104/4885PTGS2 819/4885
US-20140163045-A1 Small Molecule Xanthine Oxidase Inhibitors and Methods of Use XDH, PNPO, AOX1 XDH 1/4885KDM4E 3104/4885PTGS2 819/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.