Water

Water

SCHEMBL36578

O.O=Cc1cc(O)c(O)c(O)c1

nearest known ligand 0.94

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ABCC9ABL1ACEACHEACVR1ADORA1ADORA2AADORA2BADORA3ADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3AGTR1ALOX5ATP4AATP4BBCRBTKCACNA1ACACNA1BCACNA1CCACNA1DCACNA1ECACNA1FCACNA1GCACNA1HCACNA1ICACNA1SCACNA2D1CACNA2D2CACNA2D3CACNA2D4CACNB1CACNB2CACNB3CACNB4CACNG1CACNG2CACNG3CACNG4CACNG5CACNG6CACNG7CACNG8CALCRLCFBCHRM1CHRM2CHRM3CHRM4CHRM5CHRNA1CHRNB1CHRNDCHRNECHRNGCRBNCUL4ACXCR1CXCR2DDB1DDCDHFRDPP4DRD2DRD3DRD4EGFRERBB2ERBB4ESR1ESR2FDPSFKBP1AFLT1FLT3FLT4GARTGHSRGRIA1GRIA2GRIA3GRIA4GRIK1GRIK2GRIK3GRIK4GRIK5GRIN2AGSK3AGSK3BHDAC1HDAC10HDAC11HDAC2HDAC3HDAC4HDAC5HDAC6HDAC7HDAC8HDAC9HRH1HTR1AHTR1BHTR1DHTR1EHTR1FHTR2AHTR2BHTR2CHTR3AHTR3BHTR3CHTR3DHTR3EHTR4HTR5AHTR6HTR7IDH1IDH2IMPA1ITGA2BITGB3JAK1JAK2JAK3KCNJ11KCNK3KCNK9KDRKITMEN1METMMP1MMP13MMP7MMP8NANOD2NS5bODC1OPG057OPRD1OPRK1OPRM1PPARP1PARP2PDE3APDE3BPDE4APDE4BPDE4CPDE4DPDGFRBPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PKLRPPARDPPATPTGS1PTGS2RBX1ROCK1ROCK2RRM1RRM2RRM2BSCN10ASCN11ASCN1ASCN2ASCN3ASCN4ASCN5ASCN7ASCN8ASCN9ASCNN1ASCNN1BSCNN1GSIGMAR1SLC10A2SLC5A2SLC6A2SLC6A3SLC6A4SLC9A3SYKTACR1THRATHRBTOP1TUBA1ATUBA1BTUBA1CTUBA3CTUBA3ETUBA4ATUBBTUBB1TUBB2ATUBB2BTUBB3TUBB4ATUBB4BTUBB6TUBB8TYK2TYMSVDRampCblablaT-3blaT-4blaT-5blaT-6blaUOE-1dacAdacBdacCfolAfolPftsIgyrAgyrBileSmecAmrcAmrcBmrdAparCparEpbp2pbp4pbpApbpFrplArplBrplCrplDrplErplFrplIrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmE2rpmFrpmGrpmG1rpmG2rpmG3rpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUthyAykgMykgO

The experimentally established mechanism targets of Water. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTGS2 known ✓ P35354 2/20 0.54
MEN1 known ✓ O00255 2/20 0.48
EGFR known ✓ P00533 1/20 0.48
DPP4 known ✓ P27487 1/20 0.40
XDH P47989 1/20 0.57
KDM4E B2RXH2 4/20 0.54
RAB9A P51151 1/20 0.54
MAPT P10636 3/20 0.48
TDP1 Q9NUW8 3/20 0.48
ALDH1A1 P00352 3/20 0.48
BLM P54132 2/20 0.48
KMT2A Q03164 2/20 0.48
LMNA P02545 2/20 0.48
TP53 P04637 2/20 0.48
HPGD P15428 2/20 0.48
SMN1; SMN2 Q16637 2/20 0.48
HSD17B10 Q99714 2/20 0.48
RGS12 O14924 1/20 0.48
USP2 O75604 1/20 0.48
LCK P06239 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL132439 0.97 XDH (0.59) XDHKDM4EPTGS2RAB9AMAPT
SCHEMBL27935044 0.97 XDH (0.59) XDHKDM4EPTGS2RAB9AMAPT
SCHEMBL31122716 0.94 XDH (0.57) XDHKDM4EPTGS2RAB9AMAPT
Alcohol SCHEMBL28845727 0.85 XDH (0.50) XDHKDM4EPTGS2RAB9ATDP1
Benzaldehyde SCHEMBL17963717 0.84 ALDH1A1 (0.61) XDHKDM4EPTGS2RAB9AALDH1A1
SCHEMBL30822600 0.82 XDH (0.52) XDHKDM4EPTGS2RAB9AALDH1A1
SCHEMBL1056033 0.82 XDH (0.52) XDHKDM4EPTGS2RAB9AALDH1A1
SCHEMBL1527073 0.82 XDH (0.52) XDHKDM4EPTGS2RAB9AALDH1A1
SCHEMBL299751 0.80 EGFR (0.53) XDHKDM4EPTGS2RAB9AMAPT
SCHEMBL7962088 0.80 XDH (0.50) XDHKDM4EPTGS2RAB9AALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 97 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1300486-B1 Plating bath and method for depositing a metal layer on a substrate SHIPLEY CO LLC (US) 2011-03-16 EP claimed
US-20040074778-A1 Plating bath and method for depositing a metal layer on a substrate SHIPLEY COMPANY, L.L.C. (US) 2004-04-22 US claimed
US-6652731-B2 Comprises 2,3,4-trihydroxybenzaldehyde for inhibiting consumption of plating additives; integrated circuits SHIPLEY COMPANY, L.L.C. 2003-11-25 US claimed
US-20030085132-A1 Plating bath and method for depositing a metal layer on a substrate SHIPLEY COMPANY, L.L.C. 2003-05-08 US claimed
EP-1300486-A1 Plating bath and method for depositing a metal layer on a substrate Shipley Co. L.L.C. (US) 2003-04-09 EP claimed
WO-2023209250-A1 PYRIMIDO[5,4-D]PYRIMIDINE-BASED COMPOUNDS, METHODS AND USES THEREOF UNIVERSIDADE DO MINHO (PT) 2023-11-02 WO disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
US-11117987-B2 Hydroxyaryl functionalized polymers BRIDGESTONE CORPORATION (JP) 2021-09-14 US disclosed
US-11028195-B2 Hydroxyaryl functionalized polymers BRIDGESTONE CORPORATION (JP) 2021-06-08 US disclosed
US-20190322777-A1 Hydroxyaryl Functionalized Polymers BRIDGESTONE CORPORATION (JP) 2019-10-24 US disclosed
US-20190233557-A1 Hydroxyaryl Functionalized Polymers BRIDGESTONE CORPORATION (JP) 2019-08-01 US disclosed
US-10227425-B2 Hydroxyaryl functionalized polymers BRIDGESTONE CORPORATION (JP) 2019-03-12 US disclosed
EP-1300486-A1 Plating bath and method for depositing a metal layer on a substrate Shipley Co. L.L.C. (US) 2003-04-09 EP disclosed
US-20030022923-A1 Methods for treatment of sickle cell anemia MEDINOX, INC. 2003-01-30 US disclosed
EP-1173174-A4 METHODS FOR TREATMENT OF SICKLE CELL ANEMIA MEDINOX INC (US) 2002-09-18 EP disclosed
US-6355661-B1 STABILITY OF ALDEHYDES AND PROTECTED ALDEHYDES MEDINOX, INC. 2002-03-12 US disclosed
EP-1173174-A1 METHODS FOR TREATMENT OF SICKLE CELL ANEMIA Medinox, Inc. (US) 2002-01-23 EP disclosed
US-6251927-B1 TREATING SICKLE CELL ANEMIA USING PROTECTED FORMS OF ORGANIC ALDEHYDES MEDINOX, INC. 2001-06-26 US disclosed
WO-2000062777-A1 METHODS FOR TREATMENT OF SICKLE CELL ANEMIA MEDINOX, INC. (US) 2000-10-26 WO disclosed
EP-0667245-A1 Recording sheets containing alcohols and saccharides XEROX CORPORATION (US) 1995-08-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20190322777-A1 Hydroxyaryl Functionalized Polymers HAAO, HCAR3, VCL PTGS2 1427/4885MEN1 4721/4885EGFR 3863/4885
US-11028195-B2 Hydroxyaryl functionalized polymers HAAO, HCAR3, VCL PTGS2 1552/4885MEN1 4769/4885EGFR 3989/4885
US-10227425-B2 Hydroxyaryl functionalized polymers HAAO, HCAR3, VCL PTGS2 1427/4885MEN1 4721/4885EGFR 3863/4885
US-20030022923-A1 Methods for treatment of sickle cell anemia SORD, HBG1, HBG2 PTGS2 894/4885MEN1 4307/4885EGFR 4884/4885
US-11117987-B2 Hydroxyaryl functionalized polymers HAAO, HCAR3, VCL PTGS2 1427/4885MEN1 4721/4885EGFR 3863/4885
US-20190233557-A1 Hydroxyaryl Functionalized Polymers HAAO, HCAR3, VCL PTGS2 1552/4885MEN1 4769/4885EGFR 3989/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.