SCHEMBL9252072

SCHEMBL9252072

CC(C)(C)C(=O)OCn1cnc2ccc(CN)cc2c1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNF P01375 1/20 0.43
LMNA P02545 2/20 0.41
MCL1 Q07820 1/20 0.41
MMP13 P45452 4/20 0.41
RECQL P46063 1/20 0.40
MAPK10 P53779 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
SCD O00767 3/20 0.39
TRPA1 O75762 1/20 0.39
HDAC6 Q9UBN7 2/20 0.39
HDAC3 O15379 1/20 0.39
HDAC4 P56524 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC7 Q8WUI4 1/20 0.39
HDAC2 Q92769 1/20 0.39
HDAC10 Q969S8 1/20 0.39
HDAC11 Q96DB2 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC9 Q9UKV0 1/20 0.39
HDAC5 Q9UQL6 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9253194 0.89 LMNA (0.43) TNFLMNAMCL1MMP13RECQL
SCHEMBL5565180 0.85 TNF (0.43) TNFLMNAMCL1MMP13RECQL
SCHEMBL9601170 0.85 TRPA1 (0.47) TNFLMNAMCL1SMN1; SMN2TRPA1
SCHEMBL10431213 0.82 P2RX3 (0.43) TNFLMNAMMP13RECQLMAPK10
SCHEMBL9366964 0.81 MMP13 (0.52) MMP13RECQLMAPK10SMN1; SMN2
SCHEMBL6589975 0.81 SMN1; SMN2 (0.53) LMNARECQLMAPK10SMN1; SMN2
SCHEMBL13646422 0.80 TNF (0.56) TNFLMNAMCL1SMN1; SMN2HDAC6
SCHEMBL9248248 0.79 ALDH1A1 (0.45) LMNASMN1; SMN2HDAC6HDAC3HDAC4
SCHEMBL5500566 0.78 ESR1 (0.47) TNFLMNASMN1; SMN2HDAC6
SCHEMBL6017313 0.76 HRH3 (0.39) TNFLMNAMCL1MMP13

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5395838-A Aromatic aminomethyl substitutes compounds IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1995-03-07 US disclosed
EP-0373891-B1 Anti-tumour agents ICI PLC (GB) 1994-11-02 EP disclosed
US-5252573-A Quinazoline derivatives IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1993-10-12 US disclosed
US-5089499-A Anticarcinogenic agents; thymidylate synthetase inhibitors; antiallergens; psoriasis IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1992-02-18 US disclosed
EP-0373891-A2 Anti-tumour agents IMPERIAL CHEMICAL INDUSTRIES PLC (GB) 1990-06-20 EP disclosed