SCHEMBL9252598

SCHEMBL9252598

COc1cc(C(=O)O)cc(C#N)c1OC(C)=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.51
TPMT P51580 2/20 0.50
CA12 O43570 2/20 0.47
CA1 P00915 2/20 0.47
CA2 P00918 2/20 0.47
CA4 P22748 2/20 0.47
CA6 P23280 2/20 0.47
CA7 P43166 2/20 0.47
CA9 Q16790 2/20 0.47
CA14 Q9ULX7 2/20 0.47
PKM P14618 2/20 0.47
CA3 P07451 1/20 0.47
CA5A P35218 1/20 0.47
CA5B Q9Y2D0 1/20 0.47
HPGD P15428 2/20 0.46
PTGS2 P35354 1/20 0.45
ALDH1A1 P00352 3/20 0.44
KDM4E B2RXH2 1/20 0.44
GAA P10253 1/20 0.44
RAB9A P51151 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8848303 0.91 ALDH1A1 (0.50) TSHRTPMTCA12CA1CA2
SCHEMBL668055 0.84 TSHR (0.64) TSHRTPMTCA12CA1CA2
SCHEMBL28046034 0.81 TPMT (0.49) TPMTCA12CA1CA2CA4
SCHEMBL7371883 0.80 TOP1 (0.45) TSHRALDH1A1KDM4EGAARAB9A
SCHEMBL7368999 0.78 LMNA (0.53) TSHRTPMTHPGDALDH1A1HTT
SCHEMBL15673397 0.78 TSHR (0.65) TSHRTPMTCA12CA1CA2
SCHEMBL8726199 0.76 HPGD (0.48) TSHRTPMTCA12CA1CA2
SCHEMBL7373217 0.75 TUBB4A (0.54) HPGDALDH1A1CNR2
SCHEMBL9787608 0.75 TPMT (0.60) TPMTCA12CA1CA2CA4
SCHEMBL10323635 0.74 TPMT (0.44) TPMTCA12CA1CA2CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5446194-A Pharmacologically active catechol derivatives ORION-YHTYMA OY (FI) 1995-08-29 US disclosed
US-5283352-A Transferase inhibitor ORION-YHTYMA OY (FI) 1994-02-01 US disclosed
US-5112861-A Inhibitors of catechol-methyl-transferase enzyme, levodopa ORION-YHTYMA OY (FI) 1992-05-12 US disclosed
US-4963590-A ENZYME INHIBITOR FOR TREATING PARKINSON'S DISEASE ALONG WITH DOPA;POTENTIATION ORION-YHTYMA OY (FI) 1990-10-16 US disclosed