SCHEMBL9252637

SCHEMBL9252637

COc1cccc(S(C)(=O)=O)c1OC

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.47
HTR6 P50406 1/20 0.47
MAOB P27338 1/20 0.46
CA12 O43570 3/20 0.44
CA1 P00915 3/20 0.44
CA2 P00918 3/20 0.44
CA14 Q9ULX7 3/20 0.44
NFE2L2 Q16236 3/20 0.42
PTGS1 P23219 1/20 0.41
PTGS2 P35354 1/20 0.41
CA7 P43166 2/20 0.41
CA9 Q16790 2/20 0.41
CA4 P22748 1/20 0.41
HSD11B1 P28845 1/20 0.40
EED O75530 1/20 0.40
PRMT1 Q99873 1/20 0.40
LMNA P02545 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
ODC1 P11926 1/20 0.40
NPC1 O15118 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6912891 0.86 HTR6 (0.53) SMN1; SMN2HTR6MAOBCA12CA1
SCHEMBL668439 0.84 HTR6 (0.47) SMN1; SMN2HTR6MAOBCA12CA1
SCHEMBL6968672 0.84 HTR6 (0.47) SMN1; SMN2HTR6MAOBCA12CA1
Hydrochloric Acid SCHEMBL1796557 0.82 HTR6 (0.46) SMN1; SMN2HTR6MAOBCA12CA1
SCHEMBL29969255 0.82 TRPV4 (0.49) SMN1; SMN2HTR6MAOBCA12CA1
SCHEMBL1713241 0.82 TRPV4 (0.49) SMN1; SMN2HTR6MAOBCA12CA1
SCHEMBL791503 0.82 CA2 (0.50) SMN1; SMN2HTR6CA12CA1CA2
SCHEMBL69581 0.81 HTR6 (0.62) SMN1; SMN2HTR6CA12CA1CA2
SCHEMBL30514823 0.81 HTR6 (0.62) SMN1; SMN2HTR6CA12CA1CA2
SCHEMBL3555416 0.79 L3MBTL1 (0.51) SMN1; SMN2HTR6CA12CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7919508-B2 3-piperidinylisochroman-5-ols as dopamine agonists AVENTIS PHARMACEUTICALS INC. (US) 2011-04-05 US disclosed
EP-1749001-B1 3-PIPERIDINYLISOCHROMAN-5-OLS AS DOPAMINE AGONISTS AVENTIS PHARMA INC (US) 2010-03-03 EP disclosed
US-20070099955-A1 3-PIPERIDINYLISOCHROMAN-5-OLS AS DOPAMINE AGONISTS AVENTIS PHARMACEUTICALS INC. (US) 2007-05-03 US disclosed
US-5446194-A Pharmacologically active catechol derivatives ORION-YHTYMA OY (FI) 1995-08-29 US disclosed
US-5283352-A Transferase inhibitor ORION-YHTYMA OY (FI) 1994-02-01 US disclosed
US-5112861-A Inhibitors of catechol-methyl-transferase enzyme, levodopa ORION-YHTYMA OY (FI) 1992-05-12 US disclosed
US-4963590-A ENZYME INHIBITOR FOR TREATING PARKINSON'S DISEASE ALONG WITH DOPA;POTENTIATION ORION-YHTYMA OY (FI) 1990-10-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070099955-A1 3-PIPERIDINYLISOCHROMAN-5-OLS AS DOPAMINE AGONISTS DRD3, DRD2, DRD4 SMN1; SMN2 1261/4885HTR6 118/4885MAOB 309/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.