SCHEMBL9254028

SCHEMBL9254028

N=C(N)c1ccc(-c2c[nH]c(C3CCC(CCC(=O)O)CC3)n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
DGAT1 O75907 8/20 0.45
ITGB3 P05106 9/20 0.43
ITGA2B P08514 9/20 0.43
ITGB2 P05107 1/20 0.36
ITGAM P11215 1/20 0.36
CYP2C9 P11712 1/20 0.36
F10 P00742 1/20 0.36
PRSS1 P07477 1/20 0.36
PRSS2 P07478 1/20 0.36
PRSS3 P35030 1/20 0.36
ST14 Q9Y5Y6 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9259393 0.88 ITGB3 (0.39) DGAT1ITGB3ITGA2BCYP2C9F10
SCHEMBL9258178 0.81 ITGB3 (0.46) ITGB3ITGA2BF10PRSS1PRSS2
SCHEMBL9053167 0.77 ACHE (0.41) DGAT1ITGB3ITGA2B
SCHEMBL9053164 0.77 ACHE (0.41) DGAT1ITGB3ITGA2B
SCHEMBL9250975 0.73 FFAR1 (0.40) DGAT1
SCHEMBL9254802 0.72 ITGB3 (0.42) ITGB3ITGA2BPRSS1
SCHEMBL8949275 0.70 ITGB3 (0.46) ITGB3ITGA2BF10PRSS1PRSS2
SCHEMBL9259330 0.70 ITGB3 (0.42) ITGB3ITGA2BF10PRSS1PRSS2
SCHEMBL9256974 0.70 ITGB3 (0.51) ITGB3ITGA2BF10PRSS1PRSS2
SCHEMBL9253132 0.70 ITGB3 (0.51) ITGB3ITGA2BF10PRSS1PRSS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed