SCHEMBL9250975

SCHEMBL9250975

NC1CCC(c2nc(-c3ccc(CCC(=O)O)cc3)c[nH]2)CC1

nearest known ligand 0.40

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
FFAR1 O14842 6/20 0.40
SYK P43405 1/20 0.40
FFAR4 Q5NUL3 6/20 0.39
HRH3 Q9Y5N1 1/20 0.37
S1PR1 P21453 1/20 0.36
S1PR3 Q99500 1/20 0.36
S1PR5 Q9H228 1/20 0.36
DGAT1 O75907 1/20 0.35
CA1 P00915 1/20 0.35
CA2 P00918 1/20 0.35
F2 P00734 1/20 0.35
KEAP1 Q14145 1/20 0.35
SPHK1 Q9NYA1 1/20 0.34
RXRA P19793 1/20 0.34
RXRB P28702 1/20 0.34
RXRG P48443 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9247113 0.87 HRH3 (0.42) SYKHRH3SPHK1
SCHEMBL9254028 0.73 DGAT1 (0.45) DGAT1
Hydrochloric Acid SCHEMBL9408096 0.70 ITGB3 (0.51) FFAR1FFAR4HRH3
SCHEMBL408754 0.70 NPC1 (0.55)
SCHEMBL442390 0.70 NPC1 (0.55)
SCHEMBL6488402 0.69 FFAR1 (0.57) FFAR1FFAR4CA1CA2KEAP1
SCHEMBL9256974 0.68 ITGB3 (0.51) FFAR1F2
SCHEMBL9253132 0.68 ITGB3 (0.51) FFAR1F2
SCHEMBL15824768 0.68 PTGS1 (0.43)
SCHEMBL1725663 0.68 METAP2 (0.37)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed