SCHEMBL9254462

SCHEMBL9254462

NCc1ccc(-c2ccc(-n3cnc(CCC(=O)O)c3)nn2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDK1 Q15118 4/20 0.38
FFAR1 O14842 5/20 0.33
LOXL2 Q9Y4K0 1/20 0.33
ACACB O00763 1/20 0.32
CPB1 P15086 2/20 0.32
CPB2 Q96IY4 2/20 0.32
FFAR4 Q5NUL3 1/20 0.32
P4HTM Q9NXG6 1/20 0.31
MAP4K4 O95819 1/20 0.31
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
NFKB1 P19838 1/20 0.31
NFKB2 Q00653 1/20 0.31
RELA Q04206 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
TBXAS1 P24557 1/20 0.30
PDK2 Q15119 1/20 0.30
PDK3 Q15120 1/20 0.30
PDK4 Q16654 1/20 0.30
NR1H4 Q96RI1 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9257352 0.86 PDK1 (0.36) PDK1LOXL2ACACBCPB1CPB2
SCHEMBL9568440 0.85 ITGB3 (0.39) PDK1MAP4K4
SCHEMBL9568572 0.83 PDK1 (0.39) PDK1CPB1CPB2
Hydrochloric Acid SCHEMBL9255416 0.82 PDK1 (0.39) PDK1CPB1CPB2
SCHEMBL9247446 0.81 PDK1 (0.35) PDK1ACACBCPB1CPB2
SCHEMBL9251800 0.80 PDK1 (0.36) PDK1FFAR1ACACBNPC1RAB9A
SCHEMBL9253978 0.79 ITGB3 (0.37) PDK1MAP4K4
SCHEMBL9254123 0.77 CPB1 (0.37) PDK1LOXL2ACACBCPB1CPB2
SCHEMBL9246913 0.76 GCG (0.38) PDK1NPC1RAB9ANFKB1NFKB2
SCHEMBL8863938 0.73 TMPRSS15 (0.36) PDK1MAP4K4NPC1RAB9ASMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed