SCHEMBL9568440

SCHEMBL9568440

N=C(N)c1ccc(-c2ccc(-n3cnc(CCC(=O)O)c3)nn2)cc1

nearest known ligand 0.39

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 12/20 0.39
ITGA2B P08514 12/20 0.39
PDK1 Q15118 1/20 0.35
F10 P00742 2/20 0.34
PRSS1 P07477 2/20 0.34
F2 P00734 1/20 0.34
MAP4K4 O95819 1/20 0.34
TMPRSS15 P98073 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9253978 0.94 ITGB3 (0.37) ITGB3ITGA2BPDK1F10PRSS1
SCHEMBL8863938 0.88 TMPRSS15 (0.36) ITGB3ITGA2BPDK1F10PRSS1
SCHEMBL9250967 0.87 MAP4K4 (0.41) ITGB3ITGA2BF10PRSS1F2
SCHEMBL9251800 0.87 PDK1 (0.36) PDK1
SCHEMBL9254094 0.86 F2 (0.37) ITGB3ITGA2BPDK1F10PRSS1
SCHEMBL9256993 0.85 ITGB3 (0.40) ITGB3ITGA2BF10PRSS1F2
SCHEMBL9254462 0.85 PDK1 (0.38) PDK1MAP4K4
SCHEMBL9250512 0.84 POLB (0.36) PDK1F10PRSS1F2MAP4K4
SCHEMBL9253138 0.84 F10 (0.32) PDK1F10PRSS1F2MAP4K4
SCHEMBL9257720 0.84 ITGB3 (0.33) ITGB3ITGA2BPDK1F10PRSS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP claimed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed