Bromide

Bromide

SCHEMBL9254604

Br.Br.Cn1c(-c2ccc(C(=N)N)cc2)nc2cc(C(=O)NCCC(=O)O)cnc21

nearest known ligand 0.43

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 13/20 0.43
ITGA2B P08514 13/20 0.43
NAMPT P43490 1/20 0.39
F2 P00734 3/20 0.39
F10 P00742 2/20 0.39
ITGB2 P05107 1/20 0.39
ITGAM P11215 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
SLC22A2 O15244 1/20 0.39
PLG P00747 1/20 0.39
PLAT P00750 1/20 0.39
PROC P04070 1/20 0.39
HPN P05981 1/20 0.39
PRSS1 P07477 1/20 0.39
PRSS2 P07478 1/20 0.39
NQO2 P16083 1/20 0.39
PRSS3 P35030 1/20 0.39
SLC47A2 Q86VL8 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9252486 0.99 ITGB3 (0.43) ITGB3ITGA2BNAMPTF2F10
SCHEMBL9249665 0.90 TMPRSS15 (0.42) ITGB3ITGA2BNAMPTF2F10
SCHEMBL9248776 0.87 NAMPT (0.41) ITGB3NAMPTHDAC1HDAC8HDAC6
SCHEMBL9249490 0.84 HDAC1 (0.56) ITGB3ITGA2BNAMPTF2F10
SCHEMBL9254738 0.84 ITGB3 (0.41) ITGB3ITGA2BITGB2ITGAM
SCHEMBL9252708 0.82 CHEK2 (0.51) ITGB3ITGA2BF2F10HDAC1
SCHEMBL9254049 0.81 ITGB3 (0.43) ITGB3ITGA2BF2
SCHEMBL9252571 0.81 ITGB3 (0.45) ITGB3ITGA2BNAMPTF2F10
SCHEMBL9249572 0.79 ITGB3 (0.56) ITGB3ITGA2BNAMPTF2HDAC1
SCHEMBL9247795 0.79 ITGB3 (0.44) ITGB3ITGA2BF2HDAC1HDAC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed