SCHEMBL9256882

SCHEMBL9256882

COC(=O)CCNC(=O)c1cc2nc(-c3ccc(C(=N)N)cc3)n(C)c2cc1N(C)C

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CHEK2 O96017 1/20 0.38
HDAC1 Q13547 3/20 0.38
HDAC8 Q9BY41 3/20 0.38
HDAC6 Q9UBN7 3/20 0.38
PRSS12 P56730 4/20 0.38
TMPRSS15 P98073 2/20 0.38
HDAC3 O15379 2/20 0.37
HDAC2 Q92769 2/20 0.37
ITGB3 P05106 1/20 0.36
ITGA2B P08514 1/20 0.36
NQO2 P16083 1/20 0.35
F2 P00734 3/20 0.35
PTGER4 P35408 1/20 0.35
KDM5B Q9UGL1 1/20 0.35
BRD4 O60885 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL9246087 0.92 CHEK2 (0.36) CHEK2HDAC1HDAC8HDAC6PRSS12
SCHEMBL9255526 0.91 ITGB3 (0.43) CHEK2HDAC1HDAC8HDAC6PRSS12
SCHEMBL9255062 0.89 CHEK2 (0.40) CHEK2HDAC1HDAC8HDAC6PRSS12
SCHEMBL9255533 0.88 NPC1 (0.40) CHEK2HDAC1HDAC8HDAC6PRSS12
SCHEMBL9252454 0.88 PRSS12 (0.38) CHEK2HDAC1HDAC8HDAC6PRSS12
SCHEMBL9249905 0.87 CHEK2 (0.39) CHEK2HDAC1HDAC8HDAC6PRSS12
SCHEMBL9251414 0.85 CHEK2 (0.38) CHEK2HDAC1HDAC8HDAC6PRSS12
Acetic Acid SCHEMBL9256132 0.85 CHEK2 (0.39) CHEK2HDAC1HDAC8HDAC6PRSS12
SCHEMBL8863519 0.85 HDAC1 (0.52) HDAC1HDAC8HDAC6TMPRSS15HDAC3
SCHEMBL9254880 0.85 CHEK2 (0.49) CHEK2HDAC1HDAC8HDAC6TMPRSS15

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5434150-A Anticoagulants, cardiovascular disorders DR. KARL THOMAE GMBH (DE) 1995-07-18 US disclosed
EP-0531883-A1 Condensed 5-membered ring heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-03-17 EP disclosed