SCHEMBL9258029

SCHEMBL9258029

CCCN(CCC)CC1=COc2cc(O)ccc2O1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 4/20 0.37
DRD2 P14416 3/20 0.37
DRD1 P21728 2/20 0.37
DRD4 P21917 2/20 0.37
DRD5 P21918 2/20 0.37
OPRM1 P35372 1/20 0.35
OPRD1 P41143 1/20 0.35
OPRK1 P41145 1/20 0.35
HTR1D P28221 1/20 0.35
BCHE P06276 1/20 0.34
HRH3 Q9Y5N1 1/20 0.33
HTR1A P08908 1/20 0.33
CYP3A4 P08684 2/20 0.32
CYP2D6 P10635 1/20 0.32
TSHR P16473 1/20 0.32
NFKB1 P19838 1/20 0.32
ADRA1D P25100 1/20 0.32
ADRA1A P35348 1/20 0.32
ADRA1B P35368 1/20 0.32
HIF1A Q16665 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9263496 0.77 NR1H2 (0.39) DRD3DRD2OPRM1OPRD1OPRK1
SCHEMBL9258362 0.72 HPGD (0.43) DRD3OPRM1OPRD1OPRK1TSHR
SCHEMBL4243799 0.70 CYP3A4 (0.43) CYP3A4HSD17B10ESR2KDM4E
SCHEMBL9258041 0.67 CYP3A4 (0.32) DRD3DRD2DRD1DRD4DRD5
SCHEMBL9255807 0.66 MAPT (0.41) DRD3DRD2OPRM1OPRD1OPRK1
SCHEMBL7098613 0.64 MTNR1A (0.40)
SCHEMBL7205599 0.64 EGFR (0.43) CYP2D6HSD17B10ESR1ESR2KDM4E
SCHEMBL8580093 0.64 CA12 (0.49) CYP2D6HSD17B10ESR1ESR2
SCHEMBL1206711 0.63 HRH3 (0.69) DRD3DRD2DRD1DRD4DRD5
SCHEMBL7021029 0.63 MTNR1A (0.51) DRD3DRD2DRD4CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5439909-A 2-Substituted with amide or thioamide group; antioxidant for lipoproteins, antilipemic agents, anticholesterol agents ADIR ET COMPAGNIE (FR) 1995-08-08 US disclosed
US-5420132-A Antilipemic agents ADIR ET COMPAGNIE (FR) 1995-05-30 US disclosed
EP-0624582-A1 Substituted benzodioxine, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1994-11-17 EP disclosed