SCHEMBL9258191

SCHEMBL9258191

CC1CC2(CCC(=O)O2)C(C)CN1C

nearest known ligand 0.43

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.33
HTT P42858 1/20 0.33
HRH3 Q9Y5N1 2/20 0.32
MEN1 O00255 1/20 0.30
OPRM1 P35372 1/20 0.30
OPRD1 P41143 1/20 0.30
KMT2A Q03164 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10147277 0.71 HSD11B1 (0.30)
SCHEMBL14278564 0.68 TSHR (0.37) LMNA
SCHEMBL1474193 0.67 TSHR (0.43) LMNAKMT2A
SCHEMBL1474192 0.67 TSHR (0.43) LMNAKMT2A
SCHEMBL9249537 0.66 LMNA (0.36) LMNAGAAHTTHRH3
SCHEMBL17995482 0.64 LMNA (0.31) LMNA
SCHEMBL13482601 0.63 LMNA (0.30) LMNA
SCHEMBL5276863 0.62 MAPK1 (0.33)
SCHEMBL10303795 0.60 PRKCA (0.39) LMNA
SCHEMBL17995472 0.60 TSHR (0.43) LMNAKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0311313-B1 Heterocyclic spiro compounds and their preparation YAMANOUCHI PHARMA CO LTD (JP) 1995-05-10 EP disclosed
US-5412096-A Treatment of senile dementia, Alzheimer*s disease, cholinergic activators YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1995-05-02 US disclosed
US-5041549-A Cholinergin agents YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1991-08-20 US disclosed
US-4996210-A Cognition activators, nervous system disorders; muscarinic acetylcholine receptor agonists; 2,8-dimethyl-3-methylene-1-oxa-8-azaspiro[4.5]decane for example YAMANOUCHI PHARMACEUTICAL CO., LTD. (JP) 1991-02-26 US disclosed
EP-0311313-A2 Heterocyclic spiro compounds and their preparation YAMANOUCHI PHARMACEUTICAL CO. LTD. (JP) 1989-04-12 EP disclosed