SCHEMBL14278564

SCHEMBL14278564

C[C@@H]1CCCC12CCC(=O)O2

nearest known ligand 0.46

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.37
LMNA P02545 1/20 0.37
PTGS2 P35354 1/20 0.34
MAPK1 P28482 2/20 0.33
CYP2C9 P11712 1/20 0.33
CA1 P00915 1/20 0.33
CA9 Q16790 1/20 0.33
MAPT P10636 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1474193 0.94 TSHR (0.43) TSHRLMNAPTGS2MAPK1CYP2C9
SCHEMBL1474192 0.94 TSHR (0.43) TSHRLMNAPTGS2MAPK1CYP2C9
SCHEMBL17995472 0.87 TSHR (0.43) TSHRLMNAMAPK1CYP2C9CA1
SCHEMBL17995479 0.77 TSHR (0.41) TSHRLMNAMAPK1CYP2C9MAPT
SCHEMBL12203799 0.72 MAPK1 (0.49) TSHRLMNAMAPK1CYP2C9MAPT
SCHEMBL17995484 0.72 TSHR (0.47) TSHRLMNAMAPK1CYP2C9MAPT
SCHEMBL16797125 0.72 TSHR (0.40) TSHRLMNAMAPK1CYP2C9MAPT
SCHEMBL10910306 0.69 PTAFR (0.33) TSHRLMNACA1CA9MAPT
SCHEMBL821890 0.68 TSHR (0.31) TSHRLMNAMAPK1CYP2C9
SCHEMBL9258191 0.68 LMNA (0.34) LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-RE44734-E1 Process for the production of 3-oxo-pregn-4-ene-21,17-carbolactones by the metal free oxidation of 17-(3-hydroxypropyl)-3,17-dihydroxyandrostanes BAYER INTELLECTUAL PROPERTY GMBH (DE) 2014-01-28 US disclosed
US-7319154-B2 Oxidation of 17 alpha -(3-hydroxypropyl)-6 beta ,7 beta ;15 beta ,16 beta -dimethylene-androstane-3 beta ,5 beta ,17 beta -triol in the presence of a catalytic amounts of a 2,2,6,6-tetramethylpiperidine-N-oxide derivative at a pH of at least 8.0 BAYER SCHERING PHARMA AG (DE) 2008-01-15 US disclosed
US-20070021603-A1 Process for the production of 3-oxo-pregn-4-ene-21,17-carbolactones by the metal free oxidation of 17-(3-hydroxypropyl)-3,17-dihydroxyandrostanes BAYER PHARMA AKTIENGESELLSCHAFT (DE) 2007-01-25 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070021603-A1 Process for the production of 3-oxo-pregn-4-ene-21,17-carbolactones by the metal free oxidation of 17-(3-hydroxypropyl)-3,17-dihydroxyandrostanes HSD17B7, HSD17B13, HSD17B3 TSHR 4505/4885LMNA 2506/4885PTGS2 179/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.