SCHEMBL9258704

SCHEMBL9258704

COC(=O)CCc1ccc(-c2nc(-c3ccc(C(=N)N)cc3)c[nH]2)cc1NC(=O)c1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.40
AAK1 Q2M2I8 1/20 0.39
F10 P00742 4/20 0.37
F2 P00734 3/20 0.37
HDAC2 Q92769 6/20 0.37
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
ITGB3 P05106 2/20 0.36
ITGA2B P08514 2/20 0.36
MAPT P10636 1/20 0.36
PRSS1 P07477 3/20 0.35
TYMS P04818 1/20 0.35
HDAC3 O15379 1/20 0.35
NR1H4 Q96RI1 1/20 0.35
CFD P00746 1/20 0.35
MAPK14 Q16539 1/20 0.35
SMO Q99835 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9254909 0.91 ITGB3 (0.45) HDAC1F10F2HDAC2NPC1
SCHEMBL9568476 0.90 TMPRSS15 (0.34) HDAC1F10F2ITGB3ITGA2B
SCHEMBL9252190 0.84 F10 (0.37) F10F2ITGB3ITGA2BPRSS1
SCHEMBL9253817 0.84 TMPRSS15 (0.38) F10F2ITGB3ITGA2BPRSS1
SCHEMBL9251429 0.84 TMPRSS15 (0.36) HDAC1F10F2ITGB3ITGA2B
SCHEMBL9250408 0.83 CHEK1 (0.38) ITGB3ITGA2BMAPT
SCHEMBL9258892 0.82 ITGB3 (0.39) F10ITGB3ITGA2BMAPTTYMS
SCHEMBL9254513 0.81 CHEK1 (0.40) ITGB3ITGA2BPRSS1
SCHEMBL9257084 0.79 F2 (0.41) HDAC1F10F2ITGB3ITGA2B
SCHEMBL9568559 0.79 F2 (0.41) HDAC1F10F2ITGB3ITGA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed