SCHEMBL9254909

SCHEMBL9254909

N=C(N)c1ccc(-c2c[nH]c(-c3ccc(CCC(=O)O)c(NC(=O)c4ccccc4)c3)n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ITGB3 P05106 2/20 0.45
ITGA2B P08514 2/20 0.45
TYMS P04818 1/20 0.42
F10 P00742 4/20 0.38
HDAC1 Q13547 5/20 0.38
HDAC2 Q92769 4/20 0.37
F2 P00734 2/20 0.37
AURKA O14965 1/20 0.37
TTK P33981 1/20 0.37
ITK Q08881 1/20 0.37
AURKB Q96GD4 1/20 0.37
INCENP Q9NQS7 1/20 0.37
HDAC3 O15379 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
PPARG P37231 1/20 0.36
PLG P00747 1/20 0.36
PLAU P00749 1/20 0.36
PLAT P00750 1/20 0.36
KLKB1 P03952 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9258704 0.91 HDAC1 (0.40) ITGB3ITGA2BTYMSF10HDAC1
SCHEMBL9258892 0.89 ITGB3 (0.39) ITGB3ITGA2BTYMSF10
SCHEMBL9253735 0.84 F10 (0.38) ITGB3ITGA2BF10F2PRSS1
SCHEMBL9254490 0.83 F10 (0.38) ITGB3ITGA2BF10
SCHEMBL9255778 0.83 ITGB3 (0.37) ITGB3ITGA2BF10PRSS1
SCHEMBL9568476 0.80 TMPRSS15 (0.34) ITGB3ITGA2BF10HDAC1F2
SCHEMBL9254911 0.79 F7 (0.37) ITGB3ITGA2BF10F2PLG
SCHEMBL9255039 0.79 S1PR1 (0.43) ITGB3ITGA2BF10PLAU
SCHEMBL9256974 0.77 ITGB3 (0.51) ITGB3ITGA2BF10F2PLG
SCHEMBL9253132 0.77 ITGB3 (0.51) ITGB3ITGA2BF10F2PLG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5463071-A Tetrazole derivatives; useful for inhibiting undesirable cell aggregation DR. KARL THOMAE GMBH (DE) 1995-10-31 US disclosed
EP-0525629-A2 5-membered heterocycles, process for their preparation and medicaments containing them Dr. Karl Thomae GmbH (DE) 1993-02-03 EP disclosed