SCHEMBL9258757

SCHEMBL9258757

COc1cccc2c1cc1n2CCC1=O

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNFRSF1A P19438 1/20 0.43
FNTA P49354 1/20 0.41
PGGT1B P53609 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
USP2 O75604 1/20 0.40
S100A4 P26447 1/20 0.40
CYP1A1 P04798 2/20 0.39
CYP1B1 Q16678 2/20 0.39
CYP1A2 P05177 1/20 0.39
PRKDC P78527 1/20 0.39
HRH4 Q9H3N8 1/20 0.37
ALDH1A1 P00352 2/20 0.36
KDM4E B2RXH2 2/20 0.36
MAPT P10636 2/20 0.36
GLA P06280 1/20 0.36
HPGD P15428 1/20 0.36
DAO P14920 1/20 0.36
CYP19A1 P11511 1/20 0.36
NQO2 P16083 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2018382 0.81 ALDH1A1 (0.41) MEN1KMT2AUSP2S100A4CYP1A1
SCHEMBL9279188 0.80 ALOX5 (0.37) USP2CYP1A2PRKDCALDH1A1KDM4E
SCHEMBL13629383 0.77 PABPC1 (0.36) MEN1KMT2AUSP2CYP1A1CYP1B1
SCHEMBL9287303 0.74 KDM4E (0.48) MEN1KMT2AUSP2ALDH1A1KDM4E
SCHEMBL24916750 0.72 HTR6 (0.39) MEN1KMT2ACYP1A2ALDH1A1MAPT
SCHEMBL6983377 0.71 KMT2A (0.50) MEN1KMT2AUSP2S100A4CYP1A1
SCHEMBL6982969 0.70 KMT2A (0.46) MEN1KMT2AUSP2S100A4CYP1A1
SCHEMBL9259549 0.69 HTR2A (0.44) KMT2ADAO
SCHEMBL9264795 0.69 KDM4E (0.56) MEN1KMT2AUSP2ALDH1A1KDM4E
SCHEMBL9261555 0.69 HTR2A (0.49) TNFRSF1AMEN1KMT2AUSP2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5428043-A Tricyclic-cyclic amines as novel cholinesterase inhibitors PFIZER INC. (US) 1995-06-27 US disclosed
EP-0441517-A2 Tricyclic amines as novel cholinesterase inhibitors PFIZER INC. (US) 1991-08-14 EP disclosed