SCHEMBL9258923

SCHEMBL9258923

Nc1cccc(C2(O)CCOCC2)c1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.38
CASP1 P29466 1/20 0.38
RECQL P46063 1/20 0.38
ALOX5 P09917 9/20 0.37
HTR1D P28221 1/20 0.37
ALDH1A1 P00352 2/20 0.36
PIK3CD O00329 1/20 0.36
CA12 O43570 1/20 0.36
CA1 P00915 1/20 0.36
CA2 P00918 1/20 0.36
CA7 P43166 1/20 0.36
CA9 Q16790 1/20 0.36
TDP1 Q9NUW8 1/20 0.36
CA14 Q9ULX7 1/20 0.36
CYP11B1 P15538 2/20 0.35
CYP11B2 P19099 2/20 0.35
PRKACA P17612 1/20 0.35
PRKACG P22612 1/20 0.35
PRKACB P22694 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15133163 0.87 CYP3A4 (0.46) CYP3A4CASP1RECQLALDH1A1CA12
SCHEMBL2718795 0.83 CYP3A4 (0.42) CYP3A4CASP1RECQLALDH1A1CA12
SCHEMBL21377671 0.83 CYP3A4 (0.42) CYP3A4CASP1RECQLALDH1A1CA12
SCHEMBL3647735 0.81 CYP3A4 (0.41) CYP3A4CASP1RECQLALDH1A1CA12
SCHEMBL6257993 0.81 CYP3A4 (0.41) CYP3A4CASP1RECQLALDH1A1CA12
SCHEMBL9219871 0.80 OPRD1 (0.44) CYP3A4ALOX5HTR1DALDH1A1CA12
SCHEMBL1193696 0.79 OPRM1 (0.52) ALOX5HTR1DOPRM1OPRD1OPRK1
SCHEMBL932071 0.79 CHRNA1 (0.42) ALOX5HTR1DALDH1A1OPRM1OPRD1
SCHEMBL9429709 0.79 ALOX5 (0.37) ALOX5HTR1DCYP11B1CYP11B2HRH3
SCHEMBL1598578 0.79 ALOX5 (0.37) ALOX5HTR1DCYP11B1CYP11B2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2221051-A1 AMINE DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONIST ACTIVITY AND USE THEREOF Shionogi&Co., Ltd. (JP) 2010-08-25 EP disclosed
EP-2014285-B1 NPYY5 antagonists SHIONOGI & CO (JP) 2010-05-05 EP disclosed
EP-2017261-A1 AMINE DERIVATIVE HAVING NPY Y5 RECEPTOR ANTAGONIST ACTIVITY SHIONOGI & CO., LTD. (JP) 2009-01-21 EP disclosed
US-5432194-A Antiallergens, antinflammatory agents ABBOTT LABORATORIES (US) 1995-07-11 US disclosed
WO-1994026264-A1 (4-ALKOXYPYRAN-4-YL) SUBSTITUTED ARYLALKYLARYL-, ARYLALKENYLARYL-, AND ARYLALKYNYLARYLUREA INHIBITORS OF 5-LIPOXYGENASE ABBOTT LABORATORIES (US) 1994-11-24 WO disclosed
US-5346914-A Antiallergens, antiinflammatory agents ABBOTT LABORATORIES (US) 1994-09-13 US disclosed