SCHEMBL9259048

SCHEMBL9259048

Oc1cccc(Cl)c1C(F)(F)F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.50
ALDH1A1 P00352 4/20 0.48
NOTUM Q6P988 4/20 0.42
LMNA P02545 3/20 0.36
EGFR P00533 2/20 0.36
CA2 P00918 2/20 0.36
FYN P06241 2/20 0.36
MMP9 P14780 2/20 0.36
HPGD P15428 2/20 0.36
ALOX15 P16050 2/20 0.36
RECQL P46063 2/20 0.36
HSD17B10 Q99714 2/20 0.36
TDP1 Q9NUW8 2/20 0.36
ADAMTS4 O75173 1/20 0.36
CA1 P00915 1/20 0.36
MMP2 P08253 1/20 0.36
MMP8 P22894 1/20 0.36
CA6 P23280 1/20 0.36
CDK2 P24941 1/20 0.36
MMP12 P39900 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8722602 0.83 NOTUM (0.50) TSHRALDH1A1NOTUMLMNATDP1
SCHEMBL5512574 0.83 TDP1 (0.45) TSHRALDH1A1LMNAEGFRCA2
SCHEMBL2499899 0.77 TSHR (0.50) TSHRALDH1A1LMNAEGFRCA2
SCHEMBL1041749 0.74 NOTUM (0.43) TSHRALDH1A1NOTUMLMNAHSD17B10
SCHEMBL4891656 0.74 HSD17B1 (0.41) TSHRALDH1A1LMNAEGFRCA2
SCHEMBL4120536 0.74 ALDH1A1 (0.38) ALDH1A1LMNAEGFRCA2FYN
SCHEMBL936662 0.74 NOTUM (0.43) TSHRALDH1A1NOTUMLMNACYP1A2
SCHEMBL30368333 0.74 ALDH1A1 (0.38) ALDH1A1LMNAEGFRCA2FYN
SCHEMBL22969778 0.74 NOTUM (0.43) TSHRALDH1A1NOTUMLMNATDP1
SCHEMBL29449840 0.74 NOTUM (0.43) TSHRALDH1A1NOTUMLMNACYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 20 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116655456-A Method for efficiently purifying and separating 2-chloro-4-trifluoromethyl phenol 上虞颖泰精细化工有限公司 2023-08-29 CN claimed
CN-117510497-A DGK zeta inhibitors 山东轩竹医药科技有限公司 2024-02-06 CN disclosed
US-20230348415-A1 BISPECIFIC ANTAGONISTS OF RETINOL-BINDING PROTEIN 4 THAT STABILIZE TRANSTHYRETIN TETRAMERS, THEIR PREPARATION, AND USE IN THE TREATMENT OF COMMON AGE-RELATED COMORBIDITIES THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2023-11-02 US disclosed
CN-116655456-A Method for efficiently purifying and separating 2-chloro-4-trifluoromethyl phenol 上虞颖泰精细化工有限公司 2023-08-29 CN disclosed
CN-116507613-A Bispecific antagonists of retinol binding protein 4 which stabilize transthyretin tetramer, their preparation and use in the treatment of common age-related complications 纽约哥伦比亚大学理事会 2023-07-28 CN disclosed
EP-4181909-A2 BISPECIFIC ANTAGONISTS OF RETINOL-BINDING PROTEIN 4 THAT STABILIZE TRANSTHYRETIN TETRAMERS, THEIR PREPARATION, AND USE IN THE TREATMENT OF COMMON AGE-RELATED COMORBIDITIES The Trustees Of Columbia University In The City Of New York (US) 2023-05-24 EP disclosed
WO-2022020305-A2 BISPECIFIC ANTAGONISTS OF RETINOL-BINDING PROTEIN 4 THAT STABILIZE TRANSTHYRETIN TETRAMERS, THEIR PREPARATION, AND USE IN THE TREATMENT OF COMMON AGE-RELATED COMORBIDITIES THE TRUSTEES OF COLUMBIA UNIVERSITY IN THE CITY OF NEW YORK (US) 2022-01-27 WO disclosed
US-5382686-A Process for preparing nitrodiphenyl (thio) ethers BAYER AKTIENGESELLSCHAFT (DE) 1995-01-17 US disclosed
EP-0304725-B1 PROCESS FOR THE PREPARATION OF NITRO-DIPHENYL(THIO) ETHERS BAYER AG (DE) 1992-01-22 EP disclosed
EP-0298803-B1 PROCESS FOR THE PERHALOALKYLATION OF AROMATIC DERIVATIVES RHONE-POULENC CHIMIE (FR) 1991-09-04 EP disclosed
EP-0206951-B1 PROCESS FOR THE PERFLUOROALKYLATION OF AROMATIC DERIVATIVES RHONE-POULENC CHIMIE (FR) 1990-03-21 EP disclosed
EP-0304725-A1 Process for the preparation of nitro-diphenyl(thio) ethers BAYER AG (DE) 1989-03-01 EP disclosed
EP-0298803-A1 Process for the perhaloalkylation of aromatic derivatives RHONE-POULENC CHIMIE (FR) 1989-01-11 EP disclosed
US-4731450-A Process for perfluoroalkylation of aromatic derivatives RHONE-POULENC SPECIALITES CHIMIQUES (FR) 1988-03-15 US disclosed
US-4704483-A FLUORINATION WITH POTASSIUM FLUORIDE OCCIDENTAL CHEMICAL CORPORATION (US) 1987-11-03 US disclosed
EP-0206951-A2 Process for the perfluoroalkylation of aromatic derivatives RHONE-POULENC CHIMIE (FR) 1986-12-30 EP disclosed
US-4582948-A VAPOR PHASE CHLORO-DENITRATION REACTION OCCIDENTAL CHEMICAL CORPORATION (US) 1986-04-15 US disclosed
EP-0159388-A2 Preparation of nuclear chlorinated compounds OCCIDENTAL CHEMICAL CORPORATION (US) 1985-10-30 EP disclosed
US-4504689-A Process for the preparation of phenates substituted by halogen groups or of the corresponding phenols RHONE-POULENC AGROCHIMIE (FR) 1985-03-12 US disclosed
US-4470930-A Preparation of nuclear chlorinated aromatic compounds OCCIDENTAL CHEMICAL CORPORATION (US) 1984-09-11 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230348415-A1 BISPECIFIC ANTAGONISTS OF RETINOL-BINDING PROTEIN 4 THAT STABILIZE TRANSTHYRETIN TETRAMERS, THEIR PREPARATION, AND USE IN THE TREATMENT OF COMMON AGE-RELATED COMORBIDITIES TTR, RBP4, RBP1 TSHR 19/4885ALDH1A1 2655/4885NOTUM 3184/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.