SCHEMBL9268354

SCHEMBL9268354

CSc1ccc(Oc2ccc(-c3c(C)[nH]c(C)cc3=O)cc2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SLC2A1 P11166 1/20 0.44
HPGD P15428 4/20 0.35
ALDH1A1 P00352 4/20 0.35
SLC6A4 P31645 4/20 0.35
GSK3B P49841 1/20 0.34
GSTP1 P09211 1/20 0.34
PTGS2 P35354 4/20 0.34
TSHR P16473 3/20 0.34
HSD17B10 Q99714 3/20 0.34
CYP1A2 P05177 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2C9 P11712 1/20 0.34
ALOX15 P16050 1/20 0.34
NFKB1 P19838 1/20 0.34
PDE4A P27815 1/20 0.34
BLM P54132 1/20 0.34
PMP22 Q01453 1/20 0.34
PDE4B Q07343 1/20 0.34
PDE4C Q08493 1/20 0.34
PDE4D Q08499 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9265637 0.84 GSTP1 (0.51) SLC2A1GSTP1TSHRCYP1A2CYP3A4
SCHEMBL9268241 0.83 SLC2A1 (0.63) SLC2A1HPGDPTGS2TSHRCYP1A2
SCHEMBL9262847 0.80 PTGS2 (0.44) SLC2A1PTGS2KDM4E
SCHEMBL9267476 0.80 MAPT (0.46) SLC2A1PTGS2MAPTRAB9A
SCHEMBL9454898 0.79 ALDH1A1 (0.51) HPGDALDH1A1PTGS2ATMKDM4E
SCHEMBL9455121 0.75 ALDH1A1 (0.46) HPGDALDH1A1PTGS2CYP1A2KDM4E
SCHEMBL9255564 0.75 ACHE (0.41) HPGDALDH1A1PTGS2KDM4EGAA
SCHEMBL9267616 0.75 SLC2A1 (0.39) SLC2A1GSTP1PTGS2KDM4E
SCHEMBL9455077 0.72 KEAP1 (0.49) PTGS2KDM4EMAPTMEN1KMT2A
SCHEMBL9269889 0.72 PDGFRA (0.49) HPGDALDH1A1PTGS2HSD17B10CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5403934-A Heterocyclic compounds BURROUGHS WELLCOME CO. (US) 1995-04-04 US disclosed
WO-1991013873-A1 HETEROCYCLIC COMPOUNDS THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-19 WO disclosed
EP-0447164-A1 Heterocyclic compounds THE WELLCOME FOUNDATION LIMITED (GB) 1991-09-18 EP disclosed