SCHEMBL9268753

SCHEMBL9268753

C[CH]c1ccc(N(C)C(=O)OCc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.50
MAPT P10636 1/20 0.50
HPGD P15428 1/20 0.50
CHRNB2 P17787 1/20 0.45
CHRNB4 P30926 1/20 0.45
CHRNA3 P32297 1/20 0.45
CHRNA4 P43681 1/20 0.45
AKR1B10 O60218 2/20 0.43
AKR1B1 P15121 2/20 0.43
CA12 O43570 1/20 0.43
CA4 P22748 1/20 0.43
CA6 P23280 1/20 0.43
CA5A P35218 1/20 0.43
CA7 P43166 1/20 0.43
CA9 Q16790 1/20 0.43
CA14 Q9ULX7 1/20 0.43
CA5B Q9Y2D0 1/20 0.43
LMNA P02545 1/20 0.43
HCAR2 Q8TDS4 1/20 0.42
CTDSP1 Q9GZU7 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27558112 0.86 CHRNB2 (0.56) ALDH1A1MAPTHPGDCHRNB2CHRNB4
SCHEMBL12835337 0.85 ALDH1A1 (0.55) ALDH1A1MAPTHPGDCHRNB2CHRNB4
SCHEMBL12173013 0.84 ALDH1A1 (0.54) ALDH1A1MAPTHPGDCHRNB2CHRNB4
SCHEMBL5582815 0.82 ALDH1A1 (0.60) ALDH1A1MAPTHPGDCHRNB2CHRNB4
SCHEMBL5700875 0.82 ALDH1A1 (0.52) ALDH1A1MAPTHPGDCHRNB2CHRNB4
SCHEMBL5858822 0.81 ALDH1A1 (0.51) ALDH1A1MAPTHPGDCHRNB2CHRNB4
SCHEMBL10685331 0.80 ALDH1A1 (0.57) ALDH1A1MAPTHPGDCHRNB2CHRNB4
SCHEMBL19918329 0.80 ALDH1A1 (0.57) ALDH1A1MAPTHPGDCHRNB2CHRNB4
SCHEMBL7296240 0.80 ALDH1A1 (0.50) ALDH1A1MAPTHPGDCHRNB2CHRNB4
SCHEMBL5700803 0.79 LMNA (0.53) ALDH1A1MAPTHPGDCHRNB2CHRNB4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0666846-A4 1995-09-20 EP disclosed
EP-0666846-A1 NEW SUBSTITUTED AZETIDINONES AS ANTI-INFLAMMATORY AND ANTIDEGENERATIVE AGENTS MERCK & CO. INC. (US) 1995-08-16 EP disclosed