Icopezil

Icopezil

SCHEMBL9276199

O=C(O)/C=C\C(=O)O.O=C(O)C(F)(F)F.O=C1Cc2cc3c(CCC4CCN(Cc5ccccc5)CC4)noc3cc2N1

nearest known ligand 0.93

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2BTKCACNA1CCACNA1DCACNA1FCACNA1SCCR5CPT1BCPT2DPP4DRD1DRD2EGFRERBB2ERBB4HRH1HRH3HTR1AHTR2AHTR2BHTR2CHTR4JAK1JAK2JAK3MPLMTORPPIK3CAPIK3CBPIK3CDPIK3CGPIK3R1PIK3R2PIK3R3PIK3R5PPARGSLC6A2SLC6A3SLC6A4SMOTYK2pol

The experimentally established mechanism targets of Icopezil. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ACHE P22303 20/20 0.93
BCHE P06276 9/20 0.93

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Icopezil SCHEMBL9276204 1.00 ACHE (0.93) ACHEBCHE
Icopezil SCHEMBL3339253 0.96 ACHE (1.00) ACHEBCHE
Icopezil SCHEMBL2231222 0.96 ACHE (1.00) ACHEBCHE
Icopezil SCHEMBL194482 0.91 ACHE (1.00) ACHEBCHE
SCHEMBL4512593 0.87 ACHE (1.00) ACHEBCHE
SCHEMBL2402320 0.86 ACHE (0.90) ACHEBCHE
Maleic Acid SCHEMBL3926936 0.84 ACHE (0.77) ACHEBCHE
SCHEMBL220485 0.83 ACHE (1.00) ACHEBCHE
SCHEMBL2405514 0.82 ACHE (0.84) ACHEBCHE
SCHEMBL2403486 0.82 ACHE (0.82) ACHEBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0646115-A1 HETEROCYCLIC-CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 1995-04-05 EP disclosed