Icopezil

Icopezil

SCHEMBL194482

O=C1Cc2cc3c(CCC4CCN(Cc5ccccc5)CC4)noc3cc2N1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Predicted protein targets (top 2)

geneUniProtsupporting neighboursconfidence
ACHE P22303 20/20 1.00
BCHE P06276 7/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4512593 0.96 ACHE (1.00) ACHEBCHE
SCHEMBL2402320 0.95 ACHE (0.90) ACHEBCHE
Icopezil SCHEMBL2231222 0.94 ACHE (1.00) ACHEBCHE
Icopezil SCHEMBL3339253 0.94 ACHE (1.00) ACHEBCHE
SCHEMBL220485 0.92 ACHE (1.00) ACHEBCHE
SCHEMBL2405514 0.91 ACHE (0.84) ACHEBCHE
Icopezil SCHEMBL9276199 0.91 ACHE (0.93) ACHEBCHE
Icopezil SCHEMBL9276204 0.91 ACHE (0.93) ACHEBCHE
SCHEMBL2403486 0.91 ACHE (0.82) ACHEBCHE
SCHEMBL6198882 0.84 ACHE (0.73) ACHEBCHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 776 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4635489-A1 COMPOSITION FOR PREVENTING OR TREATING SIDE EFFECTS OF CHOLINESTERASE INHIBITORS Dr.Noah Biotech Inc. (KR) 2025-10-22 EP claimed
EP-4509120-A2 COMPOSITIONS FOR IMPROVING CELL VIABILITY AND METHODS OF USE THEREOF Amylyx Pharmaceuticals Inc. (US) 2025-02-19 EP claimed
US-12186330-B2 Compositions for improving cell viability and methods of use thereof Amylyx Pharmaceuticals Inc. (US) 2025-01-07 US claimed
US-20240423965-A1 FIXED DOSE COMBINATION OF CHOLINESTERASE INHIBITOR AND A QUATERNARY AMMONIUM ANTIMUSCARINIC AGENT TO TREAT NEURODEGENERATIVE COGNITIVE DISORDERS QAAM PHARMACEUTICALS LLC (US) 2024-12-26 US claimed
EP-4473964-A1 COMPOSITION COMPRISING BETA BLOCKER AND CHOLINESTERASE INHIBITOR FOR TREATMENT OF NEURODEGENERATIVE DISEASE Dr.Noah Biotech Inc. (KR) 2024-12-11 EP claimed
CN-118647376-A Compositions comprising a beta blocker and a cholinesterase inhibitor for the treatment of neurodegenerative diseases 诺亚博士生物科技有限公司 2024-09-13 CN claimed
WO-2024128473-A1 COMPOSITION FOR PREVENTING OR TREATING SIDE EFFECTS OF CHOLINESTERASE INHIBITORS 닥터노아바이오텍 주식회사 2024-06-20 WO claimed
US-20240148711-A1 COMPOSITION COMPRISING BETA BLOCKER AND CHOLINESTERASE INHIBITOR FOR TREATMENT OF NEURODEGENERATIVE DISEASE DR.NOAH BIOTECH INC. (KR) 2024-05-09 US claimed
US-20240066017-A1 PREVENTION OR TREATMENT OF BRAIN DISEASE AND ADVERSE EFFECTS OF CHOLINESTERASE INHIBITORS DR. NOAH BIOTECH INC. (KR) 2024-02-29 US claimed
US-20230414575-A1 MK2 ACTIVATING COMPOUNDS FOR USE IN TREATING VASCULAR LEAK AND ENDOTHELIAL BARRIER DISORDERS AKTTYVA THERAPEUTICS INC (US) 2023-12-28 US claimed
US-20020028834-A1 Heterocyclic-cyclic amine derivatives VILLALOBOS ANABELLA (US) 2002-03-07 US claimed
US-20020016334-A1 Pharmaceutical composition for the treatment of attention deficit hyperactivity disorder (ADHD) COE JOTHAM WADSWORTH (US) 2002-02-07 US claimed
EP-1177798-A2 A pharmaceutical composition for the treatment of attention deficit hyperactivity disorder(ADHD) comprising a nicotine receptor partial agonist and anti-ADHD agent Pfizer Products Inc. (US) 2002-02-06 EP claimed
WO-2001085145-A2 A PHARMACEUTICAL COMPOSITION AND METHOD OF TREATMENT OF DISEASES OF COGNITIVE DYSFUNCTION IN A MAMMAL PFIZER PRODUCTS INC. (US) 2001-11-15 WO claimed
US-20010036949-A1 Pharmaceutical composition and method of treatment of diseases of cognitive dysfunction in a mammal PFIZER PRODUCTS INC. 2001-11-01 US claimed
CN-1285742-A Combination of active principles for treating senile dementia such as alzheimer dementia SANOFI SYNTHELABO (FR) 2001-02-28 CN claimed
EP-0976404-A2 A pharmaceutical composition for the prevention and treatment of diseases of cognitive dysfunction in a mammal Pfizer Products Inc. (US) 2000-02-02 EP claimed
JP-2659107-B2 EISAI CO LTD (JP) 1997-09-30 JP claimed
EP-0646115-A1 HETEROCYCLIC-CYCLIC AMINE DERIVATIVES Eisai Co., Ltd. (JP) 1995-04-05 EP claimed
WO-1992017475-A1 HETEROCYCLIC-CYCLIC AMINE DERIVATIVES PFIZER INC. (US) 1992-10-15 WO claimed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240148711-A1 COMPOSITION COMPRISING BETA BLOCKER AND CHOLINESTERASE INHIBITOR FOR TREATMENT OF NEURODEGENERATIVE DISEASE ACHE, BACE1, CHRNB4 ACHE 1/4885BCHE 6/4885
US-20020016334-A1 Pharmaceutical composition for the treatment of attention deficit hyperactivity disorder (ADHD) CHRNB4, CHRNA10, CHRNA7 ACHE 59/4885BCHE 211/4885
US-20240066017-A1 PREVENTION OR TREATMENT OF BRAIN DISEASE AND ADVERSE EFFECTS OF CHOLINESTERASE INHIBITORS ACHE, BCHE, CHAT ACHE 1/4885BCHE 2/4885
US-20240423965-A1 FIXED DOSE COMBINATION OF CHOLINESTERASE INHIBITOR AND A QUATERNARY AMMONIUM ANTIMUSCARINIC AGENT TO TREAT NEURODEGENERATIVE COGNITIVE DISORDERS ACHE, BCHE, CHRM1 ACHE 1/4885BCHE 2/4885
US-20020028834-A1 Heterocyclic-cyclic amine derivatives BCHE, ACHE, CHRM1 ACHE 2/4885BCHE 1/4885
US-12186330-B2 Compositions for improving cell viability and methods of use thereof HSPA9, CYP27A1, TUFM ACHE 3040/4885BCHE 531/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.