SCHEMBL928273

SCHEMBL928273

COc1ccccc1CCNC(=O)[C@@H]1Cc2ccccc2N1S(=O)(=O)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.60

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.49
TAAR1 Q96RJ0 1/20 0.46
LMNA P02545 2/20 0.45
SMN1; SMN2 Q16637 1/20 0.45
TGM2 P21980 1/20 0.44
RAB9A P51151 1/20 0.44
KMT2A Q03164 2/20 0.43
MEN1 O00255 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
HPGD P15428 1/20 0.43
MTNR1A P48039 1/20 0.42
MTNR1B P49286 1/20 0.42
RORC P51449 1/20 0.41
NAMPT P43490 1/20 0.41
ALDH1A1 P00352 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL928845 0.93 MAPT (0.45) MAPTTAAR1LMNASMN1; SMN2TGM2
SCHEMBL926558 0.91 MAPT (0.54) MAPTLMNASMN1; SMN2NAMPTALDH1A1
SCHEMBL926201 0.91 MAPT (0.44) MAPTTAAR1LMNASMN1; SMN2RORC
SCHEMBL926737 0.89 LMNA (0.46) MAPTLMNASMN1; SMN2RORCALDH1A1
SCHEMBL926976 0.88 HSD11B1 (0.46) MAPTTAAR1LMNASMN1; SMN2KMT2A
SCHEMBL926180 0.88 LMNA (0.48) MAPTLMNASMN1; SMN2TDP1HPGD
SCHEMBL927527 0.86 FKBP1A (0.48) LMNASMN1; SMN2TGM2RAB9AKMT2A
SCHEMBL926338 0.86 FKBP1A (0.49) RAB9AKMT2AMEN1ALDH1A1
SCHEMBL926834 0.84 RORC (0.50) SMN1; SMN2TGM2RORCALDH1A1
SCHEMBL926686 0.83 ESRRG (0.47) TGM2RAB9AKMT2AMEN1RORC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7872021-B2 LXR receptor modulators LABORATORIES FOURNIER S.A. (FR) 2011-01-18 US disclosed
US-20070099960-A1 LXR receptor modulators LABORATOIRES FOURNIER S.A. (FR) 2007-05-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070099960-A1 LXR receptor modulators NR1H2, NR1H3, PPARD MAPT 1687/4885TAAR1 742/4885LMNA 1809/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.