SCHEMBL926737

SCHEMBL926737

Cc1ccccc1CCNC(=O)[C@@H]1Cc2ccccc2N1S(=O)(=O)c1ccc(C(C)(C)C)cc1

nearest known ligand 0.46

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.46
HSD11B1 P28845 2/20 0.44
ALDH1A1 P00352 4/20 0.43
GAA P10253 1/20 0.43
RORC P51449 1/20 0.41
PTGER3 P43115 1/20 0.40
GLA P06280 1/20 0.40
PKM P14618 1/20 0.40
HTT P42858 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40
MAPT P10636 1/20 0.40
POLB P06746 1/20 0.39
NPSR1 Q6W5P4 1/20 0.38
MAPK1 P28482 1/20 0.38
MMP3 P08254 1/20 0.38
MMP8 P22894 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL926976 0.90 HSD11B1 (0.46) LMNAHSD11B1ALDH1A1GAARORC
SCHEMBL926180 0.90 LMNA (0.48) LMNAHSD11B1ALDH1A1RORCPTGER3
SCHEMBL927527 0.89 FKBP1A (0.48) LMNAALDH1A1RORCPTGER3GLA
SCHEMBL928273 0.89 MAPT (0.49) LMNAALDH1A1RORCSMN1; SMN2MAPT
SCHEMBL926338 0.88 FKBP1A (0.49) ALDH1A1GAANPSR1MAPK1
SCHEMBL927595 0.87 POLB (0.51) LMNAALDH1A1POLBNPSR1MAPK1
SCHEMBL926214 0.87 TGM2 (0.42) LMNAHSD11B1ALDH1A1RORCPTGER3
SCHEMBL926201 0.86 MAPT (0.44) LMNAALDH1A1RORCPTGER3GLA
SCHEMBL928845 0.86 MAPT (0.45) LMNARORCSMN1; SMN2MAPT
SCHEMBL926686 0.85 ESRRG (0.47) ALDH1A1RORCPOLBNPSR1MAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7872021-B2 LXR receptor modulators LABORATORIES FOURNIER S.A. (FR) 2011-01-18 US disclosed
US-20070099960-A1 LXR receptor modulators LABORATOIRES FOURNIER S.A. (FR) 2007-05-03 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20070099960-A1 LXR receptor modulators NR1H2, NR1H3, PPARD LMNA 1809/4885HSD11B1 78/4885ALDH1A1 2845/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.