SCHEMBL9287641

SCHEMBL9287641

[CH2]c1ccc(N2CCN(CCNC(=O)c3ccc(Cl)cc3)CC2)cc1

nearest known ligand 0.78

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 7/20 0.74
HTR1A P08908 2/20 0.69
DRD4 P21917 4/20 0.66
ALDH1A1 P00352 2/20 0.65
MAOA P21397 1/20 0.65
MAOB P27338 1/20 0.65
KCNH2 Q12809 1/20 0.65
CD274 Q9NZQ7 1/20 0.65
CYP1A2 P05177 1/20 0.62
CYP3A4 P08684 1/20 0.62
CYP2D6 P10635 1/20 0.62
MAPT P10636 1/20 0.62
PMP22 Q01453 1/20 0.62
SLC6A4 P31645 1/20 0.60
DRD3 P35462 2/20 0.59
ADRA1A P35348 1/20 0.59
POLB P06746 1/20 0.58

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10723708 0.85 ALDH1A1 (0.85) DRD2HTR1ADRD4ALDH1A1MAOA
SCHEMBL7371815 0.81 DRD2 (0.84) DRD2HTR1ADRD4SLC6A4DRD3
Moclobemide SCHEMBL49708 0.79 CD274 (1.00) HTR1AALDH1A1MAOAMAOBKCNH2
Moclobemide SCHEMBL3408310 0.79 CD274 (1.00) HTR1AALDH1A1MAOAMAOBKCNH2
SCHEMBL14329888 0.79 ALDH1A1 (0.94) HTR1AALDH1A1MAOAMAOBKCNH2
Moclobemide SCHEMBL11475483 0.78 CD274 (0.97) HTR1AALDH1A1MAOAMAOBKCNH2
SCHEMBL10756632 0.77 TMEM97 (0.72) DRD2HTR1ADRD4ALDH1A1MAOA
SCHEMBL1322020 0.77 DRD4 (1.00) DRD2HTR1ADRD4CYP1A2CYP3A4
SCHEMBL9387833 0.77 ALDH1A1 (0.74) DRD2HTR1AALDH1A1MAOAMAOB
SCHEMBL30301397 0.77 DRD2 (0.69) DRD2HTR1ADRD4CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0649419-A1 N-CYCLOALKYLPIPERAZINE DERIVATIVES, METHODS OF OBTAINING THEM AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM LES LABORATOIRES MERAM (FR) 1995-04-26 EP disclosed