SCHEMBL9301475

SCHEMBL9301475

COc1nc2nc[nH]c2c(=O)n1C

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATAD2 Q6PL18 1/20 0.46
ADORA2A P29274 6/20 0.45
PDE4A P27815 6/20 0.45
PDE4B Q07343 6/20 0.45
PDE4C Q08493 6/20 0.45
PDE4D Q08499 6/20 0.45
ADORA2B P29275 5/20 0.45
ADORA3 P0DMS8 2/20 0.45
ADORA1 P30542 2/20 0.45
PIK3CD O00329 1/20 0.45
ALPL P05186 1/20 0.45
TMIGD3 P0DMS9 1/20 0.45
CYP2C19 P33261 1/20 0.45
HIF1A Q16665 1/20 0.45
ALDH1A1 P00352 1/20 0.44
PDPK1 O15530 1/20 0.44
CYP1A2 P05177 2/20 0.41
LMNA P02545 1/20 0.41
MAPT P10636 1/20 0.41
PNP P00491 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20867 0.77 ATAD2 (0.53) ATAD2ADORA2APDE4APDE4BPDE4C
SCHEMBL9308358 0.76 ADORA2B (0.52) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL31685607 0.74 ADORA2A (0.49) ATAD2ADORA2APDE4APDE4BPDE4C
SCHEMBL31685659 0.74 ATAD2 (0.46) ATAD2ADORA2APDE4APDE4BPDE4C
SCHEMBL2115743 0.70 ALDH1A1 (0.52) ATAD2ADORA2APDE4APDE4BPDE4C
SCHEMBL31646363 0.69 ADORA2B (0.45) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL1867634 0.67 PDE4A (0.48) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL2343362 0.67 ADORA2A (0.44) ADORA2APDE4APDE4BPDE4CPDE4D
SCHEMBL8520502 0.67 PNP (0.57) ALDH1A1PNPPDE5A
SCHEMBL17025973 0.67 CHRNB2 (0.46) ADORA2BCYP2C19ALDH1A1CYP1A2MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2025133718-A1 AN EFFICIENT PROCESS FOR THE SYNTHESIS OF PARAXANTHINE FERTIS INDIA PVT. LTD. (IN) 2025-06-26 WO disclosed
US-5314890-A Treatment of asthma MALESCI ISTITUTO FARMACOBIOLOGICO S.P.A. (IT) 1994-05-24 US disclosed
EP-0531349-A1 1-7 SUBSTITUTED XANTHINE DERIVATIVES HAVING ANTIASTHMATIC ACTIVITY, THEIR SALTS PHYSIOLOGICALLY ACCEPTABLE, PHARMACEUTICAL COMPOSITION CONTAINING THEM AND PROCESS FOR THEIR PREPARATION MALESCI ISTITUTO FARMACOBIOLOGICO S.p.A. (IT) 1993-03-17 EP disclosed
WO-1991017993-A1 1-7 SUBSTITUTED XANTHINE DERIVATIVES HAVING ANTIASTHMATIC ACTIVITY, THEIR SALTS PHYSIOLOGICALLY ACCEPTABLE, PHARMACEUTICAL COMPOSITION CONTAINING THEM AND PROCESS FOR THEIR PREPARATION MALESCI ISTITUTO FARMACOBIOLOGICO S.P.A (IT) 1991-11-28 WO disclosed