SCHEMBL9301581

SCHEMBL9301581

CCOC(=O)Cc1nc2cc(F)c(N3CCN(C(=O)OC(C)(C)C)CC3)cc2n1C1CC1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.50
MAPT P10636 10/20 0.43
ALDH1A1 P00352 4/20 0.43
HPGD P15428 2/20 0.42
ALOX15 P16050 2/20 0.42
TSHR P16473 2/20 0.42
HSD17B10 Q99714 2/20 0.42
RORC P51449 1/20 0.42
KDM4E B2RXH2 1/20 0.42
POLB P06746 1/20 0.42
GAA P10253 1/20 0.42
GPR174 Q9BXC1 2/20 0.42
LMNA P02545 3/20 0.41
MAPK1 P28482 2/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
CASP1 P29466 1/20 0.41
CASP7 P55210 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.41
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9847732 0.90 HTT (0.43) HTTMAPTALDH1A1RORCKDM4E
SCHEMBL9301681 0.89 HTT (0.42) HTTMAPTRORCLMNASMN1; SMN2
SCHEMBL9301682 0.88 RORC (0.42) HTTMAPTRORCLMNASMN1; SMN2
SCHEMBL9303809 0.87 HTT (0.41) HTTMAPTALDH1A1RORCLMNA
SCHEMBL9301930 0.87 HTT (0.45) HTTMAPTALDH1A1HPGDALOX15
SCHEMBL9301471 0.85 RORC (0.41) HTTMAPTRORCLMNASMN1; SMN2
SCHEMBL9302442 0.85 RORC (0.41) HTTMAPTRORCLMNASMN1; SMN2
SCHEMBL9301590 0.84 MAPT (0.45) HTTMAPTALDH1A1RORCGPR174
SCHEMBL9301575 0.83 RORC (0.39) HTTMAPTRORCLMNASMN1; SMN2
SCHEMBL9303841 0.82 HPGD (0.35) HTTHPGDRORCGPR174OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5300516-A Muscarinic receptor antagonists PFIZER INC. (US) 1994-04-05 US disclosed
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed