SCHEMBL9303841

SCHEMBL9303841

CCOC(=O)Cc1nc2cc(F)c(N3CCCC3C(=O)OC(C)(C)C)cc2n1C1CC1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HPGD P15428 1/20 0.35
GPR174 Q9BXC1 1/20 0.34
CREBBP Q92793 1/20 0.34
ATR Q13535 1/20 0.34
ATRIP Q8WXE1 1/20 0.34
TRPV1 Q8NER1 1/20 0.34
CYP11B2 P19099 6/20 0.34
CYP11B1 P15538 5/20 0.34
HTT P42858 1/20 0.34
CYP19A1 P11511 1/20 0.34
MET P08581 1/20 0.34
ALK Q9UM73 1/20 0.34
HDAC1 Q13547 2/20 0.33
HDAC8 Q9BY41 2/20 0.33
HDAC6 Q9UBN7 2/20 0.33
RORC P51449 1/20 0.33
OPRM1 P35372 2/20 0.33
OPRK1 P41145 2/20 0.33
OGFRL1 Q5TC84 2/20 0.33
OPRD1 P41143 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9847716 0.91 HDAC1 (0.36) GPR174CREBBPATRATRIPTRPV1
SCHEMBL9301818 0.90 ATR (0.35) GPR174CREBBPATRATRIPTRPV1
SCHEMBL9301581 0.82 HTT (0.50) HPGDGPR174CYP11B2CYP11B1HTT
SCHEMBL9303690 0.82 OPRM1 (0.37) ATRATRIPTRPV1METALK
SCHEMBL9301930 0.80 HTT (0.45) HPGDGPR174CYP11B2CYP11B1HTT
SCHEMBL9847728 0.76 OGFRL1 (0.38) HPGDCYP11B2CYP11B1ALKOPRM1
SCHEMBL9847732 0.72 HTT (0.43) CYP11B2CYP11B1HTTRORCOPRM1
SCHEMBL9301681 0.71 HTT (0.42) CYP11B2CYP11B1HTTALKRORC
SCHEMBL9301682 0.70 RORC (0.42) CYP11B2CYP11B1HTTRORCOPRM1
SCHEMBL9303487 0.69 HDAC1 (0.34) GPR174ATRATRIPTRPV1HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed