SCHEMBL9301907

SCHEMBL9301907

O=C(O)C[C@H](NC(=O)OC(=O)c1ccccc1)C(=O)OC(=O)[C@H](CC(=O)O)NC(=O)OC(=O)c1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CASP1 P29466 13/20 0.46
ALDH1A1 P00352 1/20 0.42
TDP1 Q9NUW8 2/20 0.41
TSHR P16473 1/20 0.41
GAA P10253 1/20 0.40
MAPT P10636 1/20 0.40
KMT2A Q03164 2/20 0.40
MAPK1 P28482 1/20 0.40
HIF1A Q16665 1/20 0.40
SLC6A2 P23975 1/20 0.40
SLC6A3 Q01959 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4819455 0.89 GAA (0.48) CASP1ALDH1A1TSHRGAAMAPT
SCHEMBL11059105 0.89 GAA (0.48) CASP1ALDH1A1TSHRGAAMAPT
SCHEMBL20740123 0.83 CTSL (0.50) CASP1TDP1GAAMAPT
SCHEMBL20875154 0.83 CTSL (0.50) CASP1TDP1GAAMAPT
SCHEMBL7166866 0.79 CASP1 (0.66) CASP1
SCHEMBL732093 0.79 CASP1 (0.66) CASP1
SCHEMBL8085967 0.79 CASP1 (0.66) CASP1
SCHEMBL11062723 0.79 ALDH1A1 (0.55) ALDH1A1TSHRGAA
SCHEMBL4178228 0.78 MME (0.44) ALDH1A1TDP1TSHRMAPTKMT2A
SCHEMBL4182695 0.78 MME (0.44) ALDH1A1TDP1TSHRMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0334236-B1 Preparation of n-protected alpha-l-aspartyl-l-phenylalanine methyl ester MITSUI TOATSU CHEMICALS (JP) 1994-08-31 EP disclosed
US-5302743-A Reacting N-protected L-aspartic anhydride with L-phenylalanine methyl ester salt in non-aqueous solvent MITSUI TOATSU CHEMICALS, INC. (JP) 1994-04-12 US disclosed