SCHEMBL9302347

SCHEMBL9302347

CCn1c2ccc(N3CCN(C)CC3)c(F)c2n2c(=O)[nH]c(=S)cc12

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 1/20 0.35
POLB P06746 2/20 0.35
PLK1 P53350 2/20 0.35
MEN1 O00255 1/20 0.35
THRB P10828 1/20 0.35
TSHR P16473 1/20 0.35
RECQL P46063 1/20 0.35
KMT2A Q03164 1/20 0.35
HSD17B10 Q99714 1/20 0.35
ALK Q9UM73 2/20 0.35
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
DRD3 P35462 3/20 0.32
DRD2 P14416 2/20 0.32
DRD4 P21917 2/20 0.32
HTR1A P08908 1/20 0.32
HTR2A P28223 1/20 0.32
HTR2C P28335 1/20 0.32
GAA P10253 1/20 0.31
RAD52 P43351 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301938 0.70 DRD3 (0.43) POLBMEN1KMT2AALDH1A1DRD3
SCHEMBL9302026 0.61 DRD3 (0.44) POLBMEN1KMT2AALDH1A1DRD3
SCHEMBL9302904 0.60 ALDH1A1 (0.45) SMN1; SMN2POLBMEN1THRBTSHR
SCHEMBL14922282 0.57 ALDH1A1 (0.51) SMN1; SMN2POLBRECQLHSD17B10ALDH1A1
SCHEMBL2894409 0.57 ALDH1A1 (0.60) POLBRECQLKMT2AHSD17B10ALDH1A1
SCHEMBL8253234 0.56 HTR1A (0.47) TSHRKMT2AL3MBTL1DRD3DRD2
SCHEMBL13382891 0.56 DRD2 (0.53) SMN1; SMN2POLBMEN1TSHRKMT2A
SCHEMBL12714783 0.56 ALDH1A1 (0.54) POLBRECQLKMT2AHSD17B10ALDH1A1
SCHEMBL28425579 0.56 ALDH1A1 (0.54) POLBRECQLKMT2AHSD17B10ALDH1A1
SCHEMBL16514423 0.55 ALDH1A1 (0.62) POLBRECQLKMT2AHSD17B10ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed
EP-0433648-A1 Substituted pyrimidobenzimidazole derivatives F. HOFFMANN-LA ROCHE AG (CH) 1991-06-26 EP disclosed