SCHEMBL9302522

SCHEMBL9302522

CN1CCN(c2c(F)c(NCc3ccccc3)c([N+](=O)[O-])c(NC3CC3)c2F)CC1

nearest known ligand 0.47

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SIRT6 Q8N6T7 2/20 0.47
ALDH1A1 P00352 2/20 0.44
HPGD P15428 2/20 0.44
HTR6 P50406 4/20 0.41
LMNA P02545 1/20 0.39
HRH4 Q9H3N8 4/20 0.38
ACHE P22303 3/20 0.38
BCHE P06276 2/20 0.38
BACE1 P56817 2/20 0.38
MET P08581 1/20 0.37
JAK2 O60674 1/20 0.37
JAK3 P52333 1/20 0.37
PTK2 Q05397 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
PDE5A O76074 1/20 0.36
NOD2 Q9HC29 1/20 0.36
NOD1 Q9Y239 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9301506 0.81 MAPT (0.38) SIRT6ALDH1A1HTR6LMNACYP2D6
SCHEMBL8112311 0.74 MAPT (0.39) SIRT6ALDH1A1HPGDLMNACYP2D6
SCHEMBL8112070 0.72 WDR5 (0.36) SIRT6ALDH1A1HPGDCYP2D6CYP2C9
SCHEMBL22712825 0.69 SIRT6 (0.60) SIRT6ALDH1A1HTR6HRH4MET
SCHEMBL9564453 0.68 MAPT (0.48) SIRT6ALDH1A1HTR6CYP2D6CYP2C9
SCHEMBL9302543 0.66 MAPT (0.48) SIRT6ALDH1A1LMNAACHEBCHE
SCHEMBL10570306 0.66 MAPT (0.51) SIRT6ALDH1A1HTR6LMNACYP2D6
SCHEMBL9302194 0.66 ACHE (0.39) HTR6HRH4ACHEMETPDE5A
SCHEMBL3147203 0.64 SIRT6 (0.83) SIRT6ALDH1A1HTR6CYP2C9
SCHEMBL1847175 0.64 SIRT6 (1.00) SIRT6ALDH1A1HTR6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed