SCHEMBL9302194

SCHEMBL9302194

CN1CCN(c2c(F)c(NCc3ccccc3)c3nc(CC(N)=O)n(C4CC4)c3c2F)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.39
HRH4 Q9H3N8 8/20 0.38
STAT6 P42226 2/20 0.38
HRH1 P35367 2/20 0.37
PDE5A O76074 1/20 0.36
HRH2 P25021 1/20 0.36
HRH3 Q9Y5N1 1/20 0.36
HTR6 P50406 1/20 0.35
CTNNB1 P35222 1/20 0.35
TCF7L2 Q9NQB0 1/20 0.35
IKBKB O14920 1/20 0.34
AURKA O14965 1/20 0.34
CHUK O15111 1/20 0.34
MAPK13 O15264 1/20 0.34
DAPK3 O43293 1/20 0.34
PRKCG P05129 1/20 0.34
PIM1 P11309 1/20 0.34
CDK2 P24941 1/20 0.34
MARK3 P27448 1/20 0.34
AKT1 P31749 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9302110 0.83 ACHE (0.35) ACHEHRH4STAT6HRH1PDE5A
SCHEMBL9301180 0.67 HTR6 (0.36) ACHEHRH4HRH1PDE5AHRH2
SCHEMBL9302522 0.66 SIRT6 (0.47) ACHEHRH4PDE5AHTR6MET
SCHEMBL9302311 0.64 CYP11B2 (0.44) IRAK4
Hydrochloric Acid SCHEMBL9302957 0.63 CYP11B1 (0.43)
SCHEMBL9302144 0.62 GRM5 (0.39) HRH4
SCHEMBL5170379 0.57 GAA (0.47) HRH4
SCHEMBL16489514 0.56 HRH4 (0.62) ACHEHRH4HRH1PDE5AHRH2
SCHEMBL5790195 0.56 AGXT (0.61) HRH1HRH2HRH3HTR6AURKA
SCHEMBL1588414 0.56 HRH4 (0.81) ACHEHRH4HRH1HRH2HRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5283248-A Bactericides, enzyme inhibitor of DNA-gyrase in bacteria HOFFMANN-LA ROCHE INC. (US) 1994-02-01 US disclosed