SCHEMBL9302713

SCHEMBL9302713

CC(C)(C)C(=O)c1oc(-c2cccnc2)nc1C(C)(C)C

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
IKBKB O14920 1/20 0.47
ALDH1A1 P00352 6/20 0.43
HSD17B10 Q99714 6/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
F2 P00734 1/20 0.42
ELANE P08246 1/20 0.41
KDM4E B2RXH2 9/20 0.41
NPC1 O15118 5/20 0.41
RAB9A P51151 4/20 0.41
HPGD P15428 4/20 0.41
SMN1; SMN2 Q16637 3/20 0.41
CYP1A2 P05177 2/20 0.41
CYP3A4 P08684 2/20 0.41
CYP2C9 P11712 2/20 0.41
CYP2C19 P33261 2/20 0.41
TP53 P04637 2/20 0.41
CYP2D6 P10635 1/20 0.41
MAPK1 P28482 1/20 0.41
USP2 O75604 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2112745 0.73 IKBKB (0.56) IKBKBALDH1A1HSD17B10MEN1KMT2A
SCHEMBL9302720 0.71 KIF11 (0.40) IKBKBALDH1A1HSD17B10MEN1KMT2A
SCHEMBL26054630 0.68 MKNK1 (0.65) ALDH1A1NPC1RAB9ACYP1A2CYP3A4
SCHEMBL8614787 0.67 FBP1 (0.33) ALDH1A1HSD17B10MEN1KMT2AHPGD
SCHEMBL20022402 0.67 IKBKB (0.58) IKBKBALDH1A1HSD17B10MEN1KMT2A
SCHEMBL10937913 0.67 PIN1 (0.51) ALDH1A1HSD17B10KMT2AKDM4EHPGD
SCHEMBL17773156 0.66 KMO (0.67) ALDH1A1MEN1CYP1A2CYP3A4CYP2C9
SCHEMBL9424430 0.66 FBP1 (0.47) IKBKBALDH1A1HPGD
SCHEMBL9302312 0.65 KIF11 (0.49) ALDH1A1HSD17B10MEN1KMT2AKDM4E
SCHEMBL16997515 0.65 NPC1 (0.59) ALDH1A1HSD17B10KMT2AKDM4ENPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5340815-A Inhibitors of 5-lipoxygenase and/or cyclooxygenase WARNER-LAMBERT COMPANY (US) 1994-08-23 US disclosed
US-5302597-A Enzyme inhibitors WARNER-LAMBERT COMPANY (US) 1994-04-12 US disclosed
EP-0569491-A4 2-SUBSTITUTED-4,6-DI-TERTIARY-BUTYL-5-HYDROXY-1,3-PYRIMIDINES USEFUL AS ANTIINFLAMMATORY AGENTS 1993-11-24 EP disclosed
EP-0569491-A1 2-SUBSTITUTED-4,6-DI-TERTIARY-BUTYL-5-HYDROXY-1,3-PYRIMIDINES USEFUL AS ANTIINFLAMMATORY AGENTS WARNER-LAMBERT COMPANY (US) 1993-11-18 EP disclosed
US-5248682-A Inhibitors of lipoxygenase and cyclooxygenase WARNER-LAMBERT COMPANY (US) 1993-09-28 US disclosed
US-5177079-A Antiallergen, antiulcer WARNER-LAMBERT COMPANY (US) 1993-01-05 US disclosed
WO-1992013536-A1 2-SUBSTITUTED-4,6-DI-TERTIARY-BUTYL-5-HYDROXY-1,3-PYRIMIDINES USEFUL AS ANTIINFLAMMATORY AGENTS WARNER-LAMBERT COMPANY (US) 1992-08-20 WO disclosed