SCHEMBL9303598

SCHEMBL9303598

NCCn1nc(-c2ccc(Cl)c(Cl)c2Cl)c2cnccc21

nearest known ligand 0.36

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.36
CSNK1A1 P48729 1/20 0.35
CSNK1D P48730 1/20 0.35
CSNK1E P49674 1/20 0.35
CSNK1G2 P78368 1/20 0.35
CSNK1G1 Q9HCP0 1/20 0.35
ESR1 P03372 2/20 0.32
RORC P51449 1/20 0.30
MAOA P21397 4/20 0.30
MAOB P27338 4/20 0.30
ACHE P22303 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8137244 0.93 P2RX7 (0.34) P2RX7CSNK1A1CSNK1DCSNK1ECSNK1G2
Fumaric Acid SCHEMBL8142605 0.90 CSNK1A1 (0.32) P2RX7CSNK1A1CSNK1DCSNK1ECSNK1G2
Fumaric Acid SCHEMBL8142601 0.90 CSNK1A1 (0.32) P2RX7CSNK1A1CSNK1DCSNK1ECSNK1G2
SCHEMBL9304005 0.89 P2RX7 (0.38) P2RX7RORCMAOA
Fumaric Acid SCHEMBL8138799 0.84 KDM4E (0.34) P2RX7CSNK1A1CSNK1DCSNK1ECSNK1G2
Fumaric Acid SCHEMBL8138796 0.84 KDM4E (0.34) P2RX7CSNK1A1CSNK1DCSNK1ECSNK1G2
SCHEMBL8134112 0.84 CRHR1 (0.36)
SCHEMBL8134219 0.84 CDC7 (0.41) P2RX7MAOAMAOBACHE
SCHEMBL9305694 0.82 TDP1 (0.37) P2RX7ESR1
SCHEMBL8134084 0.82 HTR2A (0.43) P2RX7

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5296491-A Pyrazolo[4,3-c]pyridines and their use as serotonin reuptake inhibitors HOECHST-ROUSSEL PHARMACEUTICALS INC. (US) 1994-03-22 US claimed