SCHEMBL9304044

SCHEMBL9304044

Cc1ccc(CCN(C)CCCC2(c3ccccc3)CC(=O)NC(=O)C2)cc1

nearest known ligand 0.42

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SIGMAR1 Q99720 8/20 0.42
KCNH2 Q12809 1/20 0.39
ADAM17 P78536 1/20 0.36
CNR2 P34972 1/20 0.36
SLC6A9 P48067 1/20 0.36
SLC6A4 P31645 2/20 0.35
SLC6A2 P23975 1/20 0.35
SLC6A3 Q01959 1/20 0.35
TMEM97 Q5BJF2 1/20 0.35
THRA P10827 1/20 0.34
THRB P10828 1/20 0.34
MEN1 O00255 1/20 0.34
CYP3A4 P08684 1/20 0.34
CYP2D6 P10635 1/20 0.34
KMT2A Q03164 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9869620 0.93 SIGMAR1 (0.49) SIGMAR1SLC6A9SLC6A4SLC6A2SLC6A3
SCHEMBL9303707 0.84 SCN1A (0.38) SIGMAR1SLC6A4CYP3A4
SCHEMBL9304202 0.82 SIGMAR1 (0.46) SIGMAR1TMEM97
SCHEMBL9303673 0.81 CNR2 (0.34) SIGMAR1ADAM17CNR2TMEM97
SCHEMBL9304790 0.73 TAAR1 (0.36) SIGMAR1SLC6A4SLC6A3
SCHEMBL9304467 0.71 UTS2R (0.35) SIGMAR1ADAM17CNR2SLC6A9TMEM97
SCHEMBL9303403 0.69 SLC6A2 (0.43) SIGMAR1KCNH2SLC6A4SLC6A2SLC6A3
SCHEMBL9467170 0.66 TSHR (0.47) SLC6A4SLC6A2SLC6A3MEN1KMT2A
Hydrochloric Acid SCHEMBL11609001 0.64 SCN1A (0.59) SIGMAR1SLC6A4SLC6A2SLC6A3TMEM97
Hydrochloric Acid SCHEMBL11610444 0.64 SIGMAR1 (0.49) SIGMAR1SLC6A4SLC6A2SLC6A3TMEM97

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0505379-B1 MUSCARINIC RECEPTOR ANTAGONISTS PFIZER LTD (GB) 1994-07-20 EP disclosed
US-5300516-A Muscarinic receptor antagonists PFIZER INC. (US) 1994-04-05 US disclosed